SCHEMBL8587770

SCHEMBL8587770

NCCc1csc2c(Cl)cccc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 6/20 0.50
HTR2A P28223 3/20 0.49
MAOB P27338 2/20 0.38
PNMT P11086 2/20 0.37
CYP2A6 P11509 3/20 0.37
CYP1A2 P05177 3/20 0.36
SLC6A4 P31645 2/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2D6 P10635 2/20 0.36
LMNA P02545 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
PGR P06401 1/20 0.36
CHRM2 P08172 1/20 0.36
HTR1A P08908 1/20 0.36
ADRA2A P08913 1/20 0.36
ADORA3 P0DMS8 1/20 0.36
AR P10275 1/20 0.36
CHRM1 P11229 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8587698 0.81 MPO (0.47) TAAR1HTR2ACYP2A6CYP1A2SLC6A4
SCHEMBL4664840 0.80 CYP2A6 (0.39) HTR2APNMTCYP2A6CYP1A2SLC6A4
SCHEMBL8589058 0.79 TAAR1 (0.48) TAAR1HTR2ACYP2A6CYP1A2SLC6A4
SCHEMBL8587766 0.79 TAAR1 (0.48) TAAR1HTR2ACYP2A6CYP1A2SLC6A4
SCHEMBL3985620 0.79 CYP2A6 (0.38) HTR2APNMTCYP2A6CYP1A2SLC6A4
SCHEMBL6002962 0.79 CYP1A2 (0.38) CYP2A6CYP1A2SLC6A4CYP3A4CYP2D6
SCHEMBL2090742 0.79 CYP2A6 (0.38) HTR2APNMTCYP2A6CYP1A2SLC6A4
SCHEMBL2091808 0.78 CYP1A2 (0.34) CYP2A6CYP1A2SLC6A4CYP3A4CYP2D6
SCHEMBL73404 0.76 TAAR1 (0.53) TAAR1HTR2AADRA1AHTR6
SCHEMBL8584219 0.72 TAAR1 (0.50) TAAR1HTR2AMAOBPNMTCYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998027984-A1 METHOD OF PRODUCING ANALGESIA BY ADMINISTRATION OF 1,2,3,4-TETRAHYDROBENZO-[b]THIENO[2,3-c]PYRIDINE AND DERIVATIVES NEUREX CORPORATION (US) 1998-07-02 WO disclosed
US-4971974-A ANOREXIGENIC AGENTS, BENZO B!THIENO 2,3-C!PYRIDINE COMPOUNDS NEUREX CORPORATION (US) 1990-11-20 US disclosed