SCHEMBL6002991

SCHEMBL6002991

FC(F)(F)C(F)(F)Oc1cccc(-c2c[nH][c]n2)c1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
XDH P47989 1/20 0.40
GRM5 P41594 1/20 0.35
KCNH2 Q12809 1/20 0.34
SCN10A Q9Y5Y9 1/20 0.34
CTSS P25774 1/20 0.34
CTSK P43235 1/20 0.34
PDE10A Q9Y233 2/20 0.34
NPY5R Q15761 1/20 0.33
USP7 Q93009 1/20 0.33
DYRK1A Q13627 4/20 0.33
DHODH Q02127 2/20 0.32
ADORA2A P29274 1/20 0.32
ADORA1 P30542 1/20 0.32
PIM1 P11309 2/20 0.32
PIM3 Q86V86 2/20 0.32
ATR Q13535 1/20 0.32
PIM2 Q9P1W9 1/20 0.32
MAPT P10636 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6002382 0.83 ALDH1A1 (0.36) XDHGRM5KCNH2SCN10ACTSS
SCHEMBL6003131 0.82 NISCH (0.32) MAPT
SCHEMBL4047980 0.80 DRD1 (0.44) KCNH2MAPTSMN1; SMN2
SCHEMBL1319008 0.78 SMN1; SMN2 (0.49) DYRK1AMAPTSMN1; SMN2
SCHEMBL4045664 0.75 IDO1 (0.53) XDHCTSS
SCHEMBL6002864 0.73 NOTUM (0.34) XDHGRM5KCNH2SCN10APDE10A
SCHEMBL2093090 0.72 IDO1 (0.49) GRM5PIM1MAPTSMN1; SMN2
SCHEMBL4049981 0.71 KMO (0.40) DHODH
SCHEMBL6002994 0.70 NISCH (0.47) XDHGRM5KCNH2SCN10ANPY5R
SCHEMBL6003511 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678185-A1 2,3-DIHYDRO-6-NITROIMIDAZO [2,1-B] OXAZOLE COMPOUNDS FOR THE TREATMENT OF TUBERCULOSIS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2006-07-12 EP disclosed
WO-2005042542-A1 2,3-DIHYDRO-6-NITROIMIDAZO (2,1-B) OXAZOLE COMPOUNDS FOR THE TREATMENT OF TUBERCULOSIS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2005-05-12 WO disclosed