SCHEMBL6003090

SCHEMBL6003090

[CH2]COC(=CC)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
PTGS1 P23219 3/20 0.41
NR4A1 P22736 1/20 0.40
NR4A2 P43354 1/20 0.40
NR4A3 Q92570 1/20 0.40
ALDH1A1 P00352 1/20 0.40
MAPT P10636 1/20 0.40
PTPN1 P18031 2/20 0.40
GSK3B P49841 1/20 0.40
NQO2 P16083 1/20 0.38
PTGS2 P35354 1/20 0.38
MAOB P27338 3/20 0.38
IDO1 P14902 2/20 0.38
SRD5A2 P31213 1/20 0.37
CYP1A1 P04798 2/20 0.37
CYP1B1 Q16678 2/20 0.37
NPSR1 Q6W5P4 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2095296 0.78 CES2 (0.47) CES2CES1PTGS1NR4A1NR4A2
SCHEMBL6002521 0.75 NR1I2 (0.46) CES2CES1ALDH1A1MAPTGSK3B
SCHEMBL10980639 0.75 CES2 (0.53) CES2CES1ALDH1A1MAPTPTPN1
SCHEMBL2095768 0.70 LMNA (0.40) MAOBIDO1
SCHEMBL8377034 0.69 CYP1A1 (0.45) CES2CES1PTGS1NR4A1NR4A2
SCHEMBL8731898 0.69 CES2 (0.54) CES2CES1PTGS1NR4A1NR4A2
SCHEMBL10720895 0.68 CES2 (0.44) CES2CES1PTGS1NR4A1NR4A2
SCHEMBL10720902 0.68 CES2 (0.44) CES2CES1PTGS1NR4A1NR4A2
SCHEMBL6663947 0.68 MAPT (0.45) NR4A1NR4A2NR4A3ALDH1A1MAPT
SCHEMBL27520453 0.67 NR4A1 (0.63) CES2CES1PTGS1NR4A1NR4A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678185-A1 2,3-DIHYDRO-6-NITROIMIDAZO [2,1-B] OXAZOLE COMPOUNDS FOR THE TREATMENT OF TUBERCULOSIS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2006-07-12 EP disclosed
WO-2005042542-A1 2,3-DIHYDRO-6-NITROIMIDAZO (2,1-B) OXAZOLE COMPOUNDS FOR THE TREATMENT OF TUBERCULOSIS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2005-05-12 WO disclosed