SCHEMBL6004840

SCHEMBL6004840

Cc1cc(Oc2ccnc3ccc(C(F)(F)F)cc23)c(-c2ccccn2)nc1C

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 10/20 0.50
CBFB Q13951 1/20 0.42
KDM4E B2RXH2 1/20 0.40
NPC1 O15118 1/20 0.40
RIPK2 O43353 3/20 0.39
GAK O14976 3/20 0.39
NLK Q9UBE8 2/20 0.39
STK16 O75716 1/20 0.39
EGFR P00533 1/20 0.39
AAK1 Q2M2I8 1/20 0.39
BMP2K Q9NSY1 1/20 0.39
IRAK3 Q9Y616 1/20 0.39
KDR P35968 3/20 0.39
MAPK14 Q16539 2/20 0.39
BRAF P15056 2/20 0.38
TNNI3K Q59H18 1/20 0.38
LCK P06239 2/20 0.38
EPHB6 O15197 1/20 0.38
ABL1 P00519 1/20 0.38
EPHA1 P21709 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6004561 0.92 TGFBR1 (0.48) TGFBR1CBFBKDM4ENPC1GAK
SCHEMBL6004657 0.86 TGFBR1 (0.57) TGFBR1CBFBKDM4ENPC1
SCHEMBL6002965 0.86 TGFBR1 (0.49) TGFBR1CBFBKDM4ENPC1
SCHEMBL6005291 0.85 TGFBR1 (0.48) TGFBR1KDM4ENPC1
SCHEMBL6004307 0.85 TGFBR1 (0.52) TGFBR1KDM4ENPC1BRAF
SCHEMBL6004725 0.84 TGFBR1 (0.48) TGFBR1CBFBKDM4ENPC1RIPK2
SCHEMBL6004226 0.84 TGFBR1 (0.48) TGFBR1CBFBKDM4ENPC1AAK1
SCHEMBL6004264 0.84 TGFBR1 (0.48) TGFBR1KDM4ENPC1EGFRKMT2A
SCHEMBL6004134 0.84 KDM4E (0.52) TGFBR1CBFBKDM4ENPC1
SCHEMBL6004154 0.83 TGFBR1 (0.47) TGFBR1KDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1724268-A1 COMPOUND HAVING TGF-BETA INHIBITORY ACTIVITY AND PHARMACEUTICAL COMPOSITION CONTAINING SAME KIRIN BEER KABUSHIKI KAISHA (JP) 2006-11-22 EP disclosed