SCHEMBL6010230

SCHEMBL6010230

CCCC[C@H](NCC(C)C)C(N)=O

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CA1 P00915 4/20 0.46
CA2 P00918 4/20 0.46
EPHX1 P07099 2/20 0.40
SLC15A1 P46059 1/20 0.40
SLC1A3 P43003 1/20 0.37
SLC1A2 P43004 1/20 0.37
SLC1A1 P43005 1/20 0.37
DPP7 Q9UHL4 7/20 0.37
DPP8 Q6V1X1 5/20 0.37
DPP4 P27487 5/20 0.37
DPP9 Q86TI2 5/20 0.37
TLR8 Q9NR97 1/20 0.36
CTSK P43235 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4824672 0.98 CA1 (0.44) CA1CA2EPHX1SLC15A1SLC1A3
SCHEMBL19475787 0.82 CA2 (0.50) CA1CA2EPHX1SLC15A1SLC1A3
SCHEMBL19901822 0.80 CYP2D6 (0.38) CA1CA2EPHX1
SCHEMBL12743627 0.79 CA2 (0.47) CA1CA2EPHX1SLC15A1SLC1A3
SCHEMBL13707903 0.77 CA2 (0.48) CA1CA2EPHX1SLC15A1SLC1A3
SCHEMBL3248461 0.76 CA2 (0.52) CA1CA2EPHX1SLC15A1SLC1A3
SCHEMBL17826032 0.76 MAPT (0.44) CA1
SCHEMBL14687523 0.76 CA2 (0.52) CA1CA2EPHX1SLC15A1SLC1A3
SCHEMBL15381234 0.76 CA1 (0.38) CA1CA2SLC15A1DPP7DPP8
SCHEMBL15381235 0.76 CA1 (0.38) CA1CA2SLC15A1DPP7DPP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1656359-A2 MACROCYCLIC BETA-SECRETASE INHIBITORS FOR THE TREATMENT OF ALZHEIMER'S DISEASE Merck & Co., Inc. (US) 2006-05-17 EP disclosed
WO-2005018545-A2 MACROCYCLIC BETA-SECRETASE INHIBITORS FOR THE TREATMENT OF ALZHEIMER'S DISEASE MERCK & CO., INC. (US) 2005-03-03 WO disclosed