SCHEMBL6010270

SCHEMBL6010270

CC(C)(C)OC(=O)N[C@@H](C(Cc1ccc(Br)cc1)c1ccccc1)[C@@H](O)CCNC(=O)O

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSS P25774 9/20 0.48
CTSK P43235 8/20 0.48
CTSB P07858 2/20 0.41
CTSL P07711 1/20 0.41
CNR1 P21554 1/20 0.41
CNR2 P34972 1/20 0.41
ATM Q13315 1/20 0.41
KLK5 Q9Y337 2/20 0.40
AKT1 P31749 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6010531 0.85 UGT1A1 (0.43) CTSSCTSKCTSBCTSLCNR1
SCHEMBL6010283 0.85 UGT1A1 (0.43) CTSSCTSKCTSBCTSLCNR1
SCHEMBL2434947 0.84 CTSS (0.48) CTSSCTSKCTSBCTSLCNR1
SCHEMBL9378904 0.73 CTSS (0.41) CTSSCTSKCTSBCTSLATM
SCHEMBL6664759 0.73 ATM (0.41) CTSSCTSKCTSBCTSLCNR1
SCHEMBL6669325 0.73 ATM (0.41) CTSSCTSKCTSBCTSLATM
SCHEMBL6663482 0.73 KLK5 (0.41) CTSSCTSKCTSBCTSLATM
SCHEMBL6666632 0.71 ALDH1A1 (0.40) CTSSCTSKCTSBCTSLATM
SCHEMBL3804911 0.70 KLK5 (0.54) CTSSCTSKCTSBCTSLATM
SCHEMBL5750531 0.69 CTSS (0.58) CTSSCTSKCTSBCTSLATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1697344-A2 HIV PROTEASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 2006-09-06 EP disclosed
WO-2005058841-A2 HIV PROTEASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 2005-06-30 WO disclosed