SCHEMBL6663482

SCHEMBL6663482

CC(C)(C)OC(=O)N[C@@H](C(Cc1ccccc1)c1ccccc1)[C@@H](O)CCc1ncc(CO)s1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KLK5 Q9Y337 3/20 0.41
ATM Q13315 1/20 0.39
CTSS P25774 3/20 0.38
CTSK P43235 2/20 0.38
CTSL P07711 1/20 0.38
CTSB P07858 1/20 0.38
PTPRB P23467 1/20 0.38
ALDH1A1 P00352 2/20 0.38
MEN1 O00255 1/20 0.37
LMNA P02545 1/20 0.37
PKM P14618 1/20 0.37
HPGD P15428 1/20 0.37
ALOX15 P16050 1/20 0.37
TSHR P16473 1/20 0.37
XBP1 P17861 1/20 0.37
HTT P42858 1/20 0.37
KMT2A Q03164 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6666632 0.93 ALDH1A1 (0.40) KLK5ATMCTSSCTSKCTSL
SCHEMBL6692480 0.93 ADRB2 (0.38) KLK5ATMCTSSCTSKCTSL
SCHEMBL6668504 0.92 ALDH1A1 (0.39) KLK5ATMCTSSCTSKCTSL
SCHEMBL6666961 0.92 ALDH1A1 (0.39) KLK5ATMCTSSCTSKCTSL
SCHEMBL6664868 0.91 CTSK (0.41) KLK5ATMCTSKALDH1A1
SCHEMBL9378904 0.89 CTSS (0.41) KLK5ATMCTSSCTSKCTSL
SCHEMBL9379291 0.87 ATM (0.39) KLK5ATMCTSSCTSKCTSL
SCHEMBL9373974 0.87 PTPRB (0.39) KLK5ATMCTSSCTSKCTSL
SCHEMBL9373933 0.86 CTSK (0.39) KLK5ATMCTSSCTSKCTSL
SCHEMBL9372986 0.86 ATM (0.38) KLK5ATMCTSSCTSKCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1450795-A1 PEPTIDE ISOSTERES CONTAINING A HETEROCYCLE USEFUL IN THE TREATMENT OF ALZHEIMER'S DISEASE Elan Pharmaceuticals, Inc. (US) 2004-09-01 EP disclosed
WO-2003047576-A1 PEPTIDE ISOSTERES CONTAINING A HETEROCYCLE USEFUL IN THE TREATMENT OF ALZHEIMER'S DISEASE ELAN PHARMACEUTICALS, INC. (US) 2003-06-12 WO disclosed
EP-0603309-A1 PEPTIDE ISOTERS CONTAINING A HETEROCYCLE AS H.I.V. INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 1994-06-29 EP disclosed