Bicarbonate

Bicarbonate

SCHEMBL6013940

NCCNCCNCO.O=C(O)O

nearest known ligand 0.55

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 5/20 0.55
CA6 P23280 5/20 0.55
CA7 P43166 5/20 0.55
CA9 Q16790 5/20 0.55
CA14 Q9ULX7 5/20 0.55
CA5B Q9Y2D0 5/20 0.55
CA2 P00918 4/20 0.55
CA4 P22748 4/20 0.55
CA5A P35218 4/20 0.55
LMNA P02545 3/20 0.55
CA3 P07451 3/20 0.55
ALOX15 P16050 3/20 0.55
TDP1 Q9NUW8 2/20 0.55
CA1 P00915 2/20 0.55
ALDH1A1 P00352 2/20 0.55
TP53 P04637 1/20 0.55
KDM4E B2RXH2 1/20 0.52
KMT2A Q03164 3/20 0.50
MEN1 O00255 2/20 0.50
RECQL P46063 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10885036 0.89 CA12 (0.69) CA12CA6CA7CA9CA14
SCHEMBL2058092 0.89 CA12 (0.69) CA12CA6CA7CA9CA14
Trientine SCHEMBL20639324 0.89 CA12 (0.69) CA12CA6CA7CA9CA14
SCHEMBL1627711 0.89
Bicarbonate SCHEMBL10634656 0.89 CA12 (0.69) CA12CA6CA7CA9CA14
Hydrochloric Acid SCHEMBL2436614 0.87 KDM4E (0.71) CA12CA6CA7CA9CA14
Hydrochloric Acid SCHEMBL27595077 0.87 KDM4E (0.71) CA12CA6CA7CA9CA14
Bicarbonate SCHEMBL2443699 0.87 CA12 (0.67) CA12CA6CA7CA9CA14
Acetic Acid SCHEMBL971104 0.85 CA12 (0.43) CA12CA6CA7CA9CA14
SCHEMBL125862 0.84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7147837-B2 Bioactivated diagnostic imaging constrast agents EPIX PHARMACEUTICALS, INC. (US) 2006-12-12 US disclosed
US-20060275216-A1 Bioactivated diagnostic imaging contrast agents EPIX PHARMACEUTICALS, INC., A DELAWARE CORPORATION 2006-12-07 US disclosed
US-20040156785-A1 Bioactivated diagnostic imaging constrast agents EPIX MEDICAL , INC., A DELAWARE CORPORATION 2004-08-12 US disclosed
EP-0907379-B1 BIOACTIVATED DIAGNOSTIC IMAGING CONTRAST AGENTS EPIX MEDICAL INC (US) 2004-06-02 EP disclosed
US-6709646-B2 MAGNETIC RESONANCE IMAGING EPIX MEDICAL, INC. 2004-03-23 US disclosed
CN-1108824-C Bioactivated diagnostic imaging contrast agents EPIX MEDICAL INC (US) 2003-05-21 CN disclosed
US-20020034476-A1 Bioactivated diagnostic imaging contrast agents EPIX MEDICAL, INC. 2002-03-21 US disclosed
CN-1215341-A Bioactivated diagnostic imaging contrast agents EPIX MEDICAL INC (US) 1999-04-28 CN disclosed
EP-0907379-A2 BIOACTIVATED DIAGNOSTIC IMAGING CONTRAST AGENTS Epix Medical, Inc. (US) 1999-04-14 EP disclosed
WO-1997036619-A2 BIOACTIVATED DIAGNOSTIC IMAGING CONTRAST AGENTS EPIX MEDICAL, INC. (US) 1997-10-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060275216-A1 Bioactivated diagnostic imaging contrast agents SMPD1, PDE7A, PDE6C CA12 172/4885CA6 284/4885CA7 41/4885
US-20020034476-A1 Bioactivated diagnostic imaging contrast agents SMPD1, SMPD4, SMPD3 CA12 316/4885CA6 378/4885CA7 30/4885
US-20040156785-A1 Bioactivated diagnostic imaging constrast agents GUCY1A2, PDE3B, PDE2A CA12 201/4885CA6 662/4885CA7 126/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.