SCHEMBL6015750

SCHEMBL6015750

CCN(CC)CC(=O)c1c[nH]c2[c]cccc12

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.52
KMT2A Q03164 5/20 0.49
MEN1 O00255 4/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
GABRA1 P14867 1/20 0.39
GABRB2 P47870 1/20 0.39
MAPT P10636 5/20 0.38
KDM4E B2RXH2 3/20 0.38
AGTR1 P30556 1/20 0.38
LMNA P02545 3/20 0.38
HTT P42858 2/20 0.38
HPGD P15428 2/20 0.36
HSD17B10 Q99714 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CTNNB1 P35222 3/20 0.35
WNT3A P56704 3/20 0.35
ADAM17 P78536 1/20 0.34
CFTR P13569 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6015920 0.86 ALDH1A1 (0.39) ALDH1A1KMT2AMEN1CYP1A2CYP2C9
SCHEMBL6015984 0.74 ALDH1A1 (0.59) ALDH1A1KMT2AMEN1CYP2C19MAPT
SCHEMBL3871239 0.73 ATM (0.54) ALDH1A1KMT2AGABRA1GABRB2MAPT
SCHEMBL6015923 0.72 KMT2A (0.62) ALDH1A1KMT2AMEN1CYP1A2CYP2C9
SCHEMBL6016007 0.72 SMN1; SMN2 (0.40) ALDH1A1KMT2AMEN1MAPTKDM4E
SCHEMBL6015634 0.72 KMT2A (0.49) ALDH1A1KMT2AMEN1MAPTLMNA
SCHEMBL6016069 0.71 KMT2A (0.64) ALDH1A1KMT2AMEN1CYP1A2CYP2C9
SCHEMBL6015996 0.69 ALDH1A1 (0.50) ALDH1A1KMT2AMEN1MAPTKDM4E
SCHEMBL6015749 0.69 KMT2A (0.51) ALDH1A1KMT2AMEN1MAPTLMNA
SCHEMBL6015793 0.66 KMT2A (0.46) ALDH1A1KMT2AMEN1CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7049312-B1 Benzothiazinone and benzoxazinone compounds ABBOTT GMBH & CO. KG (DE) 2006-05-23 US claimed
EP-1181282-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2002-02-27 EP claimed
WO-2000075139-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2000-12-14 WO claimed
US-7049312-B1 Benzothiazinone and benzoxazinone compounds ABBOTT GMBH & CO. KG (DE) 2006-05-23 US disclosed