SCHEMBL6015758

SCHEMBL6015758

Cc1[c]c2cc(N)ccc2[nH]1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.46
KEAP1 Q14145 1/20 0.46
ALDH1A1 P00352 5/20 0.37
CASP1 P29466 2/20 0.35
PSMB8 P28062 1/20 0.35
KDM4E B2RXH2 4/20 0.33
MAPT P10636 4/20 0.33
MEN1 O00255 3/20 0.33
RAB9A P51151 3/20 0.33
KMT2A Q03164 3/20 0.33
HPGD P15428 3/20 0.33
GAA P10253 3/20 0.33
PARP1 P09874 2/20 0.33
CYP3A4 P08684 1/20 0.33
TSHR P16473 1/20 0.33
MAPKAPK2 P49137 1/20 0.33
RPS6KA3 P51812 1/20 0.33
CSNK2A1 P68400 1/20 0.33
PLK3 Q9H4B4 1/20 0.33
PDE10A Q9Y233 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2071518 0.79 CA12 (0.38) KEAP1ALDH1A1PSMB8KDM4EMAPT
SCHEMBL2073264 0.76 KIF11 (0.41) KEAP1ALDH1A1KDM4EMAPTMEN1
SCHEMBL1492708 0.76 LMNA (0.42) ALDH1A1PSMB8KDM4EMAPTMEN1
SCHEMBL2073232 0.76 GAA (0.38) ALDH1A1KDM4EMEN1KMT2AHPGD
SCHEMBL2072959 0.73 KIF11 (0.43) ALDH1A1MAPTMEN1KMT2AHPGD
SCHEMBL2072922 0.73 AR (0.36) ALDH1A1CASP1KDM4EMAPTGAA
SCHEMBL2071613 0.73 KIF11 (0.40) CYP2A6ALDH1A1KDM4EMAPTMEN1
SCHEMBL2074318 0.73 KDM4E (0.50) ALDH1A1PSMB8KDM4EMAPTMEN1
SCHEMBL1435832 0.72 IMPDH2 (0.41) CYP2A6ALDH1A1MEN1KMT2AIMPDH2
SCHEMBL29547 0.70 AHR (0.37) ALDH1A1PSMB8KDM4EMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7049312-B1 Benzothiazinone and benzoxazinone compounds ABBOTT GMBH & CO. KG (DE) 2006-05-23 US claimed
CN-1636005-A Benzothiazinone and benzoxazinone compounds KNOLL AG (DE) 2005-07-06 CN claimed
EP-1181282-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2002-02-27 EP claimed
WO-2000075139-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2000-12-14 WO claimed
US-7049312-B1 Benzothiazinone and benzoxazinone compounds ABBOTT GMBH & CO. KG (DE) 2006-05-23 US disclosed
CN-1636005-A Benzothiazinone and benzoxazinone compounds KNOLL AG (DE) 2005-07-06 CN disclosed