SCHEMBL6015855

SCHEMBL6015855

CCN(CC)C(=O)COc1ccc2[c]c[nH]c2n1

nearest known ligand 0.41

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.40
KDM4E B2RXH2 1/20 0.39
GAA P10253 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
BCHE P06276 1/20 0.36
ACHE P22303 1/20 0.36
ALDH1A1 P00352 1/20 0.35
TRPM8 Q7Z2W7 8/20 0.35
HPGD P15428 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6015939 0.73 NPC1 (0.49) TSHRKDM4EGAATDP1NPC1
SCHEMBL6015867 0.71 TSHR (0.53) TSHRKDM4EGAATDP1NPC1
SCHEMBL8749756 0.62 NPC1 (0.62) TSHRKDM4EGAATDP1NPC1
SCHEMBL8749753 0.61 RAB9A (0.54) TSHRKDM4EGAATDP1NPC1
SCHEMBL10013763 0.61 NPC1 (0.81) TSHRNPC1RAB9AALDH1A1TRPM8
SCHEMBL6292262 0.61 NPC1 (0.56) TSHRKDM4EGAATDP1NPC1
SCHEMBL10682606 0.60 LTB4R (0.58) TSHRKDM4ENPC1RAB9AALDH1A1
SCHEMBL5483907 0.60 TSHR (0.63) TSHRKDM4EGAATDP1NPC1
SCHEMBL11608373 0.60 KDM4E (0.56) TSHRKDM4EGAATDP1NPC1
SCHEMBL23358696 0.59 POLB (0.69) NPC1RAB9ATRPM8SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7049312-B1 Benzothiazinone and benzoxazinone compounds ABBOTT GMBH & CO. KG (DE) 2006-05-23 US claimed
EP-1181282-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2002-02-27 EP claimed
WO-2000075139-A2 BENZOTHIAZINONE AND BENZOXAZINONE COMPOUNDS BASF AKTIENGESELLSCHAFT (DE) 2000-12-14 WO claimed
US-7049312-B1 Benzothiazinone and benzoxazinone compounds ABBOTT GMBH & CO. KG (DE) 2006-05-23 US disclosed