SCHEMBL6016347

SCHEMBL6016347

O=C(O)c1cnc(N2CCN(CCO)CC2)nc1-c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.54
KDM4E B2RXH2 4/20 0.54
MEN1 O00255 3/20 0.54
KMT2A Q03164 3/20 0.54
USP2 O75604 2/20 0.54
CASP1 P29466 2/20 0.54
CASP7 P55210 2/20 0.54
TP53 P04637 1/20 0.54
MAPT P10636 1/20 0.54
TSHR P16473 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
HTT P42858 2/20 0.52
PTPN11 Q06124 2/20 0.48
ACHE P22303 2/20 0.47
LMNA P02545 1/20 0.47
SCN9A Q15858 1/20 0.47
HTR1A P08908 1/20 0.43
CYP1A2 P05177 1/20 0.42
GLA P06280 1/20 0.42
HIF1A Q16665 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6016473 0.85 ALDH1A1 (0.57) ALDH1A1KDM4EMEN1KMT2AUSP2
SCHEMBL6016426 0.82 PTPN11 (0.53) ALDH1A1KDM4EMEN1KMT2ACASP1
Hydrochloric Acid SCHEMBL3866277 0.81 PTPN11 (0.52) ALDH1A1KDM4EMEN1KMT2ACASP1
SCHEMBL6016519 0.80 PTPN11 (0.57) ALDH1A1KDM4EMEN1KMT2AUSP2
SCHEMBL6016398 0.80 ALDH1A1 (0.55) ALDH1A1KDM4EMEN1KMT2AUSP2
SCHEMBL4112958 0.75 ALDH1A1 (0.53) ALDH1A1KDM4EKMT2AUSP2CASP1
SCHEMBL11159169 0.73 MEN1 (0.60) ALDH1A1KDM4EMEN1KMT2AUSP2
SCHEMBL6016324 0.72 CHRM5 (0.46) ALDH1A1KDM4EMEN1KMT2AMAPT
SCHEMBL6016377 0.72 PTPN11 (0.47) ALDH1A1MEN1KMT2AMAPTSMN1; SMN2
SCHEMBL6016374 0.72 PTPN11 (0.47) ALDH1A1MEN1KMT2AMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1187815-B1 4-PHENYL-PYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2006-02-08 EP disclosed
CN-1166643-C 4-phenyl-pyrimidine derivatives - 2004-09-15 CN disclosed
CN-1353697-A 4-phenyl-pyrimidine derivatives HOFFMANN LA ROCHE (CH) 2002-06-12 CN disclosed
EP-1187815-A1 4-PHENYL-PYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-03-20 EP disclosed
US-6274588-B1 NEUROKININ OR SUBSTANCE P ANTAGONISTS; CENTRAL NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDES; ANTIDEPRESSANTS, ANXIOLYTIC AGENTS HOFFMANN-LA ROCHE INC. 2001-08-14 US disclosed
WO-2000073279-A1 4-PHENYL-PYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2000-12-07 WO disclosed