SCHEMBL6016519

SCHEMBL6016519

O=C(O)c1cnc(N2CCOCC2)nc1-c1ccccc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN11 Q06124 1/20 0.57
LMNA P02545 3/20 0.57
MAPT P10636 1/20 0.57
TSHR P16473 1/20 0.57
NPSR1 Q6W5P4 1/20 0.57
ALDH1A1 P00352 11/20 0.55
HSD17B10 Q99714 10/20 0.55
CASP1 P29466 9/20 0.55
CYP1A2 P05177 8/20 0.55
CASP7 P55210 8/20 0.55
CYP2C9 P11712 4/20 0.55
CYP3A4 P08684 3/20 0.55
GLA P06280 2/20 0.55
CYP2C19 P33261 1/20 0.55
USP2 O75604 4/20 0.54
HIF1A Q16665 3/20 0.54
MAPK1 P28482 2/20 0.54
PIK3CA P42336 1/20 0.54
HPGD P15428 1/20 0.54
POLB P06746 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6016337 0.89 CASP1 (0.55) PTPN11LMNATSHRALDH1A1HSD17B10
SCHEMBL6016426 0.86 PTPN11 (0.53) PTPN11LMNATSHRNPSR1ALDH1A1
SCHEMBL10327665 0.86 PIK3CA (0.56) PTPN11ALDH1A1PIK3CAPOLBKDM4E
Hydrochloric Acid SCHEMBL3866277 0.85 PTPN11 (0.52) PTPN11LMNATSHRNPSR1ALDH1A1
SCHEMBL6016398 0.84 ALDH1A1 (0.55) LMNATSHRNPSR1ALDH1A1HSD17B10
SCHEMBL6016473 0.84 ALDH1A1 (0.57) LMNAMAPTTSHRNPSR1ALDH1A1
SCHEMBL2954462 0.84 PTPN11 (0.52) PTPN11MAPTTSHRALDH1A1HSD17B10
SCHEMBL4133710 0.84 PTPN11 (0.52) PTPN11LMNAMAPTTSHRNPSR1
SCHEMBL4126042 0.84 PTPN11 (0.52) PTPN11LMNAMAPTTSHRNPSR1
SCHEMBL2948308 0.84 PTPN11 (0.52) PTPN11LMNATSHRALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1187815-B1 4-PHENYL-PYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2006-02-08 EP disclosed
EP-1187815-A1 4-PHENYL-PYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-03-20 EP disclosed
US-6274588-B1 NEUROKININ OR SUBSTANCE P ANTAGONISTS; CENTRAL NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDES; ANTIDEPRESSANTS, ANXIOLYTIC AGENTS HOFFMANN-LA ROCHE INC. 2001-08-14 US disclosed
WO-2000073279-A1 4-PHENYL-PYRIMIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2000-12-07 WO disclosed