Morpholine

Morpholine

SCHEMBL6016412

C1COCCN1.O=C(O)c1cnc(N2CCOCC2)nc1-c1ccc(F)cc1Cl

nearest known ligand 0.49

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKAB2 O43741 2/20 0.49
PRKAG1 P54619 2/20 0.49
PRKAA2 P54646 2/20 0.49
PRKAA1 Q13131 2/20 0.49
PRKAG3 Q9UGI9 2/20 0.49
PRKAG2 Q9UGJ0 2/20 0.49
PRKAB1 Q9Y478 2/20 0.49
PIK3CA P42336 7/20 0.43
TP53 P04637 1/20 0.42
THRB P10828 1/20 0.42
AOC3 Q16853 1/20 0.42
TSHR P16473 3/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
WDR5 P61964 2/20 0.41
ALDH1A1 P00352 3/20 0.40
USP2 O75604 2/20 0.40
CYP1A2 P05177 2/20 0.40
MAPK1 P28482 2/20 0.40
HSD17B10 Q99714 2/20 0.40
KMT2A Q03164 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6016446 0.94 PRKAB2 (0.52) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL6016520 0.90 ALDH1A1 (0.44) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
Piperazine SCHEMBL6016518 0.89 ALDH1A1 (0.44) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
Morpholine SCHEMBL6016373 0.86 PIK3CA (0.47) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
Methylpiperazine SCHEMBL6016589 0.85 TACR1 (0.40) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL4124843 0.83 PIK3CA (0.49) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL6016413 0.82 TACR1 (0.43) TSHRSMN1; SMN2ALDH1A1USP2CYP1A2
SCHEMBL7987933 0.82 TP53 (0.43) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL2954462 0.80 PTPN11 (0.52) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL4119980 0.79 ALDH1A1 (0.42) TP53TSHRSMN1; SMN2ALDH1A1USP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1187815-B1 4-PHENYL-PYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2006-02-08 EP disclosed
US-6274588-B1 NEUROKININ OR SUBSTANCE P ANTAGONISTS; CENTRAL NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDES; ANTIDEPRESSANTS, ANXIOLYTIC AGENTS HOFFMANN-LA ROCHE INC. 2001-08-14 US disclosed