SCHEMBL7987933

SCHEMBL7987933

O=C(ON1CCOCC1)c1cnc(N2CCOCC2)nc1-c1ccc(F)cc1Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.43
THRB P10828 1/20 0.43
AOC3 Q16853 3/20 0.42
PRKAB2 O43741 1/20 0.41
PRKAG1 P54619 1/20 0.41
PRKAA2 P54646 1/20 0.41
PRKAA1 Q13131 1/20 0.41
PRKAG3 Q9UGI9 1/20 0.41
PRKAG2 Q9UGJ0 1/20 0.41
PRKAB1 Q9Y478 1/20 0.41
WDR5 P61964 2/20 0.41
PIK3CA P42336 2/20 0.40
ABL1 P00519 2/20 0.39
BCR P11274 2/20 0.39
CNR2 P34972 2/20 0.39
ALDH1A1 P00352 3/20 0.39
KMT2A Q03164 2/20 0.39
AR P10275 1/20 0.39
BCL6 P41182 1/20 0.38
USP2 O75604 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6016446 0.87 PRKAB2 (0.52) TP53THRBAOC3PRKAB2PRKAG1
SCHEMBL6016521 0.86 ALDH1A1 (0.39) TP53ALDH1A1BCL6USP2TSHR
SCHEMBL6016375 0.86 CNR2 (0.46) AOC3PIK3CACNR2ALDH1A1TSHR
Morpholine SCHEMBL6016412 0.82 PRKAB2 (0.49) TP53THRBAOC3PRKAB2PRKAG1
SCHEMBL6016527 0.78 HTT (0.46) AOC3PIK3CACNR2ALDH1A1KMT2A
SCHEMBL6016658 0.78 PTPN11 (0.45) AOC3ABL1BCRCNR2ALDH1A1
SCHEMBL6016700 0.76 ALDH1A1 (0.39) TP53ABL1ALDH1A1USP2TSHR
SCHEMBL4124843 0.76 PIK3CA (0.49) AOC3PRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL6016520 0.75 ALDH1A1 (0.44) TP53PRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL6016413 0.75 TACR1 (0.43) ALDH1A1KMT2ABCL6USP2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6274588-B1 NEUROKININ OR SUBSTANCE P ANTAGONISTS; CENTRAL NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDES; ANTIDEPRESSANTS, ANXIOLYTIC AGENTS HOFFMANN-LA ROCHE INC. 2001-08-14 US disclosed