SCHEMBL6016547

SCHEMBL6016547

CN1CCN(c2ncc(OC(=O)N(C)Cc3cc(C(F)(F)F)cc(C(F)(F)F)c3)c(-c3ccc(F)cc3)n2)CC1

nearest known ligand 0.57

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 13/20 0.57
CENPE Q02224 1/20 0.41
USP2 O75604 5/20 0.41
ALDH1A1 P00352 5/20 0.41
CASP1 P29466 5/20 0.41
CASP7 P55210 5/20 0.41
HIF1A Q16665 5/20 0.41
CYP1A2 P05177 4/20 0.41
CYP3A4 P08684 4/20 0.41
TSHR P16473 2/20 0.41
GLA P06280 2/20 0.41
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 3/20 0.39
HSD17B10 Q99714 2/20 0.39
CYP2C9 P11712 2/20 0.39
MAPK1 P28482 2/20 0.39
PLA2G7 Q13093 1/20 0.39
LMNA P02545 1/20 0.38
TP53 P04637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6016619 0.91 TACR1 (0.47) TACR1CENPEUSP2ALDH1A1CASP1
SCHEMBL6016733 0.88 TACR1 (0.65) TACR1
SCHEMBL6016699 0.88 TACR1 (0.65) TACR1
SCHEMBL6016649 0.86 TACR1 (0.77) TACR1
SCHEMBL6016428 0.85 TACR1 (0.64) TACR1
SCHEMBL6016586 0.85 TACR1 (0.64) TACR1
SCHEMBL6016646 0.85 TACR1 (0.63) TACR1
SCHEMBL6016548 0.81 TACR1 (0.54) TACR1CYP3A4CYP2D6CYP2C9
SCHEMBL6016610 0.81 TACR1 (0.54) TACR1CYP3A4CYP2D6CYP2C9
SCHEMBL6862187 0.80 TACR1 (0.62) TACR1CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1187815-B1 4-PHENYL-PYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2006-02-08 EP claimed