SCHEMBL6017170

SCHEMBL6017170

O=C(O)Cc1c[nH]c2cc(OCc3c(C(F)(F)F)cc(-c4ccc(OC(F)(F)F)cc4)nc3CC3CC3)ccc12

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PPARD Q03181 8/20 0.38
MMP12 P39900 2/20 0.37
PPARA Q07869 6/20 0.34
S1PR1 P21453 1/20 0.34
PPARG P37231 2/20 0.33
NR1H4 Q96RI1 1/20 0.33
PTGER4 P35408 1/20 0.33
DHODH Q02127 1/20 0.33
KDM4E B2RXH2 1/20 0.33
CHRM4 P08173 1/20 0.33
PTGES O14684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6017193 0.89 PPARD (0.40) PPARDMMP12PPARAS1PR1PPARG
SCHEMBL6017244 0.86 PPARD (0.45) PPARDPPARAPPARGPTGER4KDM4E
SCHEMBL5617216 0.81 PPARD (0.40) PPARDPPARAPPARGPTGER4KDM4E
SCHEMBL6017252 0.79 PPARD (0.47) PPARDPPARAPPARG
SCHEMBL5653757 0.78 PPARD (0.41) PPARDPPARAPPARGPTGER4KDM4E
SCHEMBL5628280 0.77 PPARD (0.43) PPARDMMP12PPARAPPARGCHRM4
SCHEMBL1549780 0.76 PPARD (0.55) PPARDPPARA
SCHEMBL5617395 0.76 PPARD (0.44) PPARDPPARAPPARGPTGER4KDM4E
SCHEMBL1550371 0.75 MMP12 (0.43) PPARDMMP12DHODHCHRM4
SCHEMBL6064622 0.74 PPARD (0.38) PPARDPPARAPPARGPTGER4KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1682535-A1 HETEROARYL DERIVATIVES AS PPAR ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2006-07-26 EP disclosed
WO-2005049606-A1 HETEROARYL DERIVATIVES AS PPAR ACTIVATORS F. HOFFMANN-LA ROCHE AG (CH) 2005-06-02 WO disclosed