SCHEMBL601719

SCHEMBL601719

CCO[C@@H](Cc1ccc(OCCc2ccc(NC(=O)OC(C)(C)C)cc2)cc1)C(=O)O

nearest known ligand 0.72

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PPARG P37231 15/20 0.72
PPARA Q07869 15/20 0.72
PPARD Q03181 4/20 0.54
ITGB3 P05106 1/20 0.47
ITGA2B P08514 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5393093 1.00 PPARG (0.72) PPARGPPARAPPARDITGB3ITGA2B
SCHEMBL5386839 0.95 PPARA (0.71) PPARGPPARAPPARDITGB3ITGA2B
SCHEMBL5991816 0.91 PPARA (0.60) PPARGPPARAPPARDITGB3ITGA2B
SCHEMBL6818773 0.91 PPARA (0.60) PPARGPPARAPPARDITGB3ITGA2B
SCHEMBL5388906 0.91 PPARA (0.60) PPARGPPARAPPARDITGB3ITGA2B
SCHEMBL5991504 0.90 PPARA (0.59) PPARGPPARAPPARDITGB3ITGA2B
SCHEMBL5991875 0.89 PPARA (0.66) PPARGPPARAPPARD
SCHEMBL5992983 0.89 PPARA (0.61) PPARGPPARAPPARD
SCHEMBL5991768 0.89 PPARA (0.58) PPARGPPARAPPARDITGB3ITGA2B
SCHEMBL5991079 0.88 PPARA (0.57) PPARGPPARAPPARDITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 134 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230375561-A1 METHODS FOR IDENTIFICATION, STRATIFICATION, AND TREATMENT OF CNS DISEASES KADDURAH DAOUK RIMA F (US) 2023-11-23 US claimed
WO-2022081350-A2 METHODS FOR IDENTIFICATION, STRATIFICATION, AND TREATMENT OF CNS DISEASES DUKE UNIVERSITY (US) 2022-04-21 WO claimed
EP-1528917-B1 DOSAGE FORM COMPRISING HIGH DOSE HIGH SOLUBLE ACTIVE INGREDIENT AS MODIFIED RELEASE AND LOW DOSE ACTIVE INGREDIENT AS IMMEDIATE RELEASE TORRENT PHARMACEUTICALS LTD (IN) 2013-06-19 EP claimed
EP-1150678-B1 USE OF 3-HYDROXY-3-METHYLGLUTARYL COENZYM A REDUCTASE INHIBITORS FOR THE MANUFACTURE OF A MEDICAMENT FOR THE TREATMENT OF DIABETIC NEUROPATHY ASTRAZENECA AB (SE) 2007-07-18 EP claimed
EP-1404309-B1 A PHARMACEUTICAL COMBINATION COMPRISING EITHER (S)-2-ETHOXY-3- 4-(2- 4-METHANE SULFONYL OXYPHENYL ETHOXY) PHENYL| PROPANOIC ACID OR 3- 4- 2- (4-TERT-BUTOXY CARBONYL AMINOPHENYL) ETHOXY| PHENYL -(S)-2-ETHOXY PROPANOIC ACID AND A BIGUANIDE DRUG ASTRAZENECA AB (SE) 2006-08-23 EP claimed
US-20060173204-A1 New 3-aryl propionic acid derivatives and analogs ANDERSSON KJELL 2006-08-03 US claimed
US-20060153916-A1 Novel dosage form TORRENT PHARMACEUTICALS LIMITED (IN) 2006-07-13 US claimed
EP-1666034-A1 Pharmaceutical combination comprising a biguanide AstraZeneca AB (SE) 2006-06-07 EP claimed
US-20050209128-A1 Use of 3-hydroxy-3-methylglutaryl coenzym a reductase inhibitors for the manufacture of a medicament for the treatment of diabetic neuropathy ASTRAZENECA AB 2005-09-22 US claimed
WO-2005065639-A2 NOVEL PHARMACEUTICAL COMPOSITIONS TORRENT PHARMACEUTICALS LIMITED (IN) 2005-07-21 WO claimed
WO-2002100413-A1 A PHARMACEUTICAL COMBINATION COMPRISING EITHER (S)-2-ETHOXY-3- [4-(2-{4-METHANE SULFONYL OXYPHENYL} ETHOXY) PHENYL] PROPANOIC ACID OR 3-{4-[2-(4-TERT- BUTOXY CARBONYL AMINOPHENYL) ETHOXY] PHENYL} -(s)-2-ETHOXY PROPANOIC ACID AND A SULONYLUREA ASTRAZENECA AB (SE) 2002-12-19 WO claimed
WO-2002096453-A1 A PHARMACEUTICAL COMBINATION COMPRISING EITHER (S)-2-ETHOXY-3 [4-(2- {4-METHANE SULFONYL OXYPHENYL} ETHOXY)PHENYL] PROPANOIC ACID OR 3-{4-[2- (4-TERT-BUTOXY CARBONYLAMINO PHENYL) ETHOXY] PHENYL}-(S)-2-ETHOXY PROPANOIC ACID AND INSULIN ASTRAZENECA AB (SE) 2002-12-05 WO claimed
WO-2002096402-A1 A PHARMACEUTICAL COMBINATION COMPRISING EITHER (S)-2-ETHOXY-3- [4-(2- {4-METHANE SULFONYL OXYPHENYL} ETHOXY) PHENYL] PROPANOIC ACID OR 3-{4-[2- (4-TERT-BUTOXY CARBONYL AMINOPHENYL) ETHOXY] PHENYL} -(S)-2-ETHOXY PROPANOIC ACID AND A BIGUANIDE DRUG ASTRAZENECA AB (SE) 2002-12-05 WO claimed
JP-2002536332-A 2002-10-29 JP claimed
EP-1150678-A1 USE OF 3-HYDROXY-3-METHYLGLUTARYL COENZYM A REDUCTASE INHIBITORS FOR THE MANUFACTURE OF A MEDICAMENT FOR THE TREATMENT OF DIABETIC NEUROPATHY AstraZeneca AB (SE) 2001-11-07 EP claimed
WO-2001040166-A1 COMMINUTED FORM OF 3-{4-[2-(4-TERT-BUTOXYCARBONYLAMINOPHENYL)ETHOXY]PHENYL}-(S)-2-ETHOXY PROPANOIC ASTRAZENECA AB (SE) 2001-06-07 WO claimed
WO-2001040165-A1 CRYSTALLINE FORM OF 3-{4-[2-(4-TERT-BUTOXYCARBONYLAMINOPHENYL)ETHOXY]PHENYL}-(S)-2-ETHOXY PROPANOIC ACID ASTRAZENECA AB (SE) 2001-06-07 WO claimed
EP-1084102-A1 NEW 3-ARYL PROPIONIC ACID DERIVATIVES AND ANALOGS AstraZeneca AB (SE) 2001-03-21 EP claimed
WO-2000045818-A1 USE OF 3-HYDROXY-3-METHYLGLUTARYL COENZYM A REDUCTASE INHIBITORS FOR THE MANUFACTURE OF A MEDICAMENT FOR THE TREATMENT OF DIABETIC NEUROPATHY ASTRAZENECA AB (SE) 2000-08-10 WO claimed
WO-1999062871-A1 NEW 3-ARYL PROPIONIC ACID DERIVATIVES AND ANALOGS ASTRAZENECA AB (SE) 1999-12-09 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060173204-A1 New 3-aryl propionic acid derivatives and analogs GPR119, INSR, IRS1 PPARG 22/4885PPARA 11/4885PPARD 8/4885
US-20230375561-A1 METHODS FOR IDENTIFICATION, STRATIFICATION, AND TREATMENT OF CNS DISEASES SLC25A20, CPT2, NDUFAB1 PPARG 567/4885PPARA 787/4885PPARD 614/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.