SCHEMBL601768

SCHEMBL601768

CCCSc1cc[nH]c(=O)c1C

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.35
PDE5A O76074 1/20 0.34
MCL1 Q07820 1/20 0.34
SOAT1 P35610 1/20 0.33
ALDH1A1 P00352 3/20 0.32
MEN1 O00255 1/20 0.32
POLB P06746 1/20 0.32
KMT2A Q03164 1/20 0.32
HTT P42858 2/20 0.32
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA7 P43166 1/20 0.32
CA13 Q8N1Q1 1/20 0.32
KDM4E B2RXH2 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
GPR84 Q9NQS5 1/20 0.31
GAA P10253 1/20 0.31
PKM P14618 1/20 0.30
APLNR P35414 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL600158 0.88 CYP2C9 (0.42) PTGS2SOAT1KDM4EGPR84
SCHEMBL601383 0.79 PTGS2 (0.32) PTGS2
SCHEMBL599638 0.77 KDM4E (0.34) PTGS2ALDH1A1KDM4EPKM
SCHEMBL601673 0.75 PARP1 (0.33) ALDH1A1KDM4EGAA
SCHEMBL601804 0.73 PTGS2 (0.53) PTGS2ALDH1A1HTTPKM
SCHEMBL600457 0.73 PNP (0.32) KDM4ENPSR1
SCHEMBL17271403 0.69 ATAD2 (0.44) MCL1ALDH1A1HTTGAA
SCHEMBL10110583 0.69 GRIN2D (0.37) ALDH1A1MEN1POLBKMT2AKDM4E
SCHEMBL22171187 0.67 AR (0.38) ALDH1A1CA12CA1CA2CA7
SCHEMBL791101 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2420500-A1 PYRIDINE THIO DERIVATIVE, AND PHARMACEUTICAL COMPOSITION WHICH CONTAINS SAME AND HAS ANTI-HELICOBACTER PYLORI ACTION aRigen Pharmaceuticals, Inc. (JP) 2012-02-22 EP disclosed
US-20120041030-A1 PYRIDINE THIO DERIVATIVE, AND PHARMACEUTICAL COMPOSITION WHICH CONTAINS SAME AND HAS ANTI-HELICOBACTER PYLORI ACTION LINK GENOMICS, INC. (JP) 2012-02-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120041030-A1 PYRIDINE THIO DERIVATIVE, AND PHARMACEUTICAL COMPOSITION WHICH CONTAINS SAME AND HAS ANTI-HELICOBACTER PYLORI ACTION TPMT, TST, PTPN11 PTGS2 347/4885PDE5A 1510/4885MCL1 4091/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.