SCHEMBL6017770

SCHEMBL6017770

Cn1c(-c2ccccn2)nc(C(=O)NCc2ccc(F)c(F)c2)c(O)c1=O

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SCD O00767 1/20 0.44
PPARG P37231 2/20 0.44
S1PR3 Q99500 5/20 0.42
KCNE1 P15382 1/20 0.42
CCR1 P32246 1/20 0.42
KCNQ1 P51787 1/20 0.42
AADAT Q8N5Z0 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
ALDH1A1 P00352 1/20 0.40
MAPK1 P28482 1/20 0.40
PDPK1 O15530 3/20 0.40
NAMPT P43490 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6018991 0.89 SMN1; SMN2 (0.53) KCNE1CCR1KCNQ1SMN1; SMN2
SCHEMBL6017765 0.89 ALDH1A1 (0.41) KCNE1CCR1KCNQ1AADATSMN1; SMN2
SCHEMBL6017750 0.88 KDM4E (0.45) KCNE1CCR1KCNQ1AADATALDH1A1
SCHEMBL6017640 0.87 MEN1 (0.51)
SCHEMBL6017740 0.87 KMT2A (0.47) KCNE1CCR1KCNQ1AADATALDH1A1
SCHEMBL6017761 0.87 CNR1 (0.47)
SCHEMBL6017839 0.84 SCD (0.46) SCDKCNE1CCR1KCNQ1AADAT
SCHEMBL6017760 0.76 SMN1; SMN2 (0.57) KCNE1CCR1KCNQ1SMN1; SMN2ALDH1A1
SCHEMBL6017737 0.76 KCNE1 (0.44) SCDKCNE1CCR1KCNQ1AADAT
SCHEMBL6017739 0.76 ALDH1A1 (0.52) SMN1; SMN2ALDH1A1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20040229892-A1 Pyrimidine carboxamides; 5-hydroxy-2-(2-(1,1-Dioxo-6-[1,2]thiazinan-2-yl)-6-oxo-1,6-dihydropyrimidine-4-carboxamides; AIDS; AIDS related complex BRISTOL-MYERS SQUIBB COMPANY 2004-11-18 US claimed
US-7037908-B2 HIV integrase inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2006-05-02 US disclosed
US-20040229892-A1 Pyrimidine carboxamides; 5-hydroxy-2-(2-(1,1-Dioxo-6-[1,2]thiazinan-2-yl)-6-oxo-1,6-dihydropyrimidine-4-carboxamides; AIDS; AIDS related complex BRISTOL-MYERS SQUIBB COMPANY 2004-11-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040229892-A1 Pyrimidine carboxamides; 5-hydroxy-2-(2-(1,1-Dioxo-6-[1,2]thiazinan-2-yl)-6-oxo-1,6-dihydropyrimidine-4-carboxamides; AIDS; AIDS related complex DUT, CDK6, TYMS SCD 969/4885PPARG 3816/4885S1PR3 3262/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.