SCHEMBL6018807

SCHEMBL6018807

CN(C)C(=O)C1(C)SC=CC1c1ccc(Cl)cc1

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.35
TSHR P16473 2/20 0.35
KMT2A Q03164 3/20 0.33
TP53 P04637 2/20 0.33
MDM2 Q00987 2/20 0.33
MAPT P10636 2/20 0.33
LMNA P02545 1/20 0.33
GAA P10253 1/20 0.33
ABCC1 P33527 1/20 0.31
CES2 O00748 1/20 0.31
CES1 P23141 1/20 0.31
MEN1 O00255 1/20 0.31
CYP1A2 P05177 1/20 0.30
HPGD P15428 1/20 0.30
ALOX12 P18054 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
1,4-Dichlorobenzene SCHEMBL27657139 0.59 TSHR (0.54) TSHRMAPTLMNACES2CES1
SCHEMBL17772002 0.58 SLC9A1 (0.45) MAPK1KMT2AMAPTLMNAGAA
SCHEMBL10491406 0.57 SLC9A1 (0.44) MAPK1KMT2AMAPTLMNAGAA
Bicarbonate SCHEMBL10971534 0.57 MAPK1 (0.50) MAPK1TSHRKMT2AMAPTLMNA
SCHEMBL20076696 0.57 GAA (0.44) MAPK1KMT2AMAPTLMNAGAA
SCHEMBL10743257 0.57 SLC9A1 (0.46) MAPK1TSHRKMT2AMAPTGAA
SCHEMBL10743245 0.57 SLC9A1 (0.46) MAPK1TSHRKMT2AMAPTGAA
SCHEMBL11395709 0.57 SLC9A1 (0.44) MAPK1KMT2AMAPTLMNAGAA
SCHEMBL10743254 0.57 SLC9A1 (0.46) MAPK1TSHRKMT2AMAPTGAA
SCHEMBL3520379 0.56 HSD11B1 (0.58)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1412347-B1 PROCESS FOR THE PREPARATION OF HETEROCYCLIC PENTALENE DERIVATIVES BASELL POLYOLEFINE GMBH (DE) 2006-01-11 EP disclosed
US-6930190-B2 Process for the preparation of heterocyclic pentalene derivatives BASELL POLYOLEFINE GMBH (DE) 2005-08-16 US disclosed
EP-1412347-A1 PROCESS FOR THE PREPARATION OF HETEROCYCLIC PENTALENE DERIVATIVES Basell Polyolefine GmbH (DE) 2004-04-28 EP disclosed
WO-2003014107-A1 PROCESS FOR THE PREPARATION OF HETEROCYCLIC PENTALENE DERIVATIVES BASELL POLYOLEFINE GMBH (DE) 2003-02-20 WO disclosed