SCHEMBL6021728

SCHEMBL6021728

COC1CCN(c2ccc(N3CCN(CC4CC4)CC3)c(C3CC(C)(C)CC(C)(C)C3)c2)C1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NTSR1 P30989 3/20 0.34
IDH1 O75874 3/20 0.33
NR1H2 P55055 1/20 0.33
NR1H3 Q13133 1/20 0.33
HTR1A P08908 3/20 0.32
HTR7 P34969 3/20 0.32
TMEM97 Q5BJF2 1/20 0.32
SIGMAR1 Q99720 1/20 0.32
USP30 Q70CQ3 2/20 0.32
ADRA1D P25100 1/20 0.31
ADRA1A P35348 1/20 0.31
ADRA1B P35368 1/20 0.31
PDE10A Q9Y233 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6021727 1.00 NTSR1 (0.34) NTSR1IDH1NR1H2NR1H3HTR1A
Hydrochloric Acid SCHEMBL4860099 0.99 NTSR1 (0.33) NTSR1IDH1NR1H2NR1H3HTR1A
Hydrochloric Acid SCHEMBL4849905 0.99 NTSR1 (0.33) NTSR1IDH1NR1H2NR1H3HTR1A
Hydrochloric Acid SCHEMBL4849902 0.99 NTSR1 (0.33) NTSR1IDH1NR1H2NR1H3HTR1A
SCHEMBL6021774 0.94 OPRD1 (0.34) IDH1NR1H2NR1H3HTR1AHTR7
Hydrochloric Acid SCHEMBL4857320 0.93 OPRD1 (0.33) IDH1NR1H2NR1H3HTR1AHTR7
Hydrochloric Acid SCHEMBL4851022 0.90 TMEM97 (0.31) TMEM97SIGMAR1
Hydrochloric Acid SCHEMBL4851029 0.90 TMEM97 (0.31) TMEM97SIGMAR1
Hydrochloric Acid SCHEMBL4849873 0.88 DRD2 (0.37) NTSR1HTR1AHTR7TMEM97SIGMAR1
Hydrochloric Acid SCHEMBL4855116 0.88 DRD2 (0.37) NTSR1HTR1AHTR7TMEM97SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1698620-B1 BENZENE COMPOUNDS DISUBSTITUTED WITH CYCLIC GROUPS AT THE 1- AND 2-POSITIONS EISAI R&D MAN CO LTD (JP) 2016-09-28 EP disclosed
EP-1698620-A1 BENZENE COMPOUNDS DISUBSTITUTED WITH CYCLIC GROUPS AT THE 1- AND 2-POSITIONS Eisai Co., Ltd. (JP) 2006-09-06 EP disclosed