SCHEMBL6024132

SCHEMBL6024132

CC(=O)Oc1cc(C)ccc1Nc1c(F)cccc1Cl

nearest known ligand 0.61

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 0.61
PTGS1 P23219 3/20 0.61
ABCB11 O95342 1/20 0.61
PPARG P37231 1/20 0.61
NR1I3 Q14994 1/20 0.61
POLB P06746 2/20 0.42
GAA P10253 2/20 0.42
DHODH Q02127 2/20 0.39
PTGES O14684 1/20 0.39
LMNA P02545 1/20 0.38
FABP3 P05413 1/20 0.38
FABP4 P15090 1/20 0.38
RAB9A P51151 1/20 0.38
CLCN2 P51788 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL577110 0.86 PTGS2 (0.50) PTGS2PTGS1ABCB11PPARGNR1I3
SCHEMBL577295 0.81 PTGS2 (0.53) PTGS2PTGS1ABCB11PPARGNR1I3
SCHEMBL3884087 0.79 PTGS2 (0.68) PTGS2PTGS1ABCB11PPARGNR1I3
SCHEMBL5533958 0.78 PTGS2 (0.82) PTGS2PTGS1ABCB11PPARGNR1I3
SCHEMBL26193724 0.77 PTGS2 (0.62) PTGS2PTGS1ABCB11PPARGNR1I3
SCHEMBL5534966 0.76 PTGS2 (0.79) PTGS2PTGS1ABCB11PPARGNR1I3
SCHEMBL27595572 0.76 PTGS2 (0.64) PTGS2PTGS1ABCB11PPARGNR1I3
Lumiracoxib SCHEMBL29377334 0.76 PTGS2 (1.00) PTGS2PTGS1ABCB11PPARGNR1I3
Lumiracoxib SCHEMBL4479 0.76 PTGS2 (1.00) PTGS2PTGS1ABCB11PPARGNR1I3
Lumiracoxib SCHEMBL29475008 0.76 PTGS2 (1.00) PTGS2PTGS1ABCB11PPARGNR1I3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100516037-C Nitrooxyderivatives of cyclooxygenase-2 inhibitors NICOX SA (FR) 2009-07-22 CN disclosed
EP-1684784-A2 COMPOSITIONS OF A CYCLOOXYGENASE-2 SELECTIVE INHIBITOR AND A NEUROTROPHIC FACTOR-MODULATING AGENT FOR THE TREATMENT OF CENTRAL NERVOUS SYSTEM MEDIATED DISORDERS Pharmacia & Upjohn Company LLC (US) 2006-08-02 EP disclosed
EP-1670417-A2 COMPOSITIONS OF A CYCLOOXYGENASE-2 SELECTIVE INHIBITOR ADMINISTERED UNDER HYPOTHERMIC CONDITIONS FOR THE TREATMENT OF ISCHENIC MEDIATED CENTRAL NERVOUS SYSTEM DISORDERS OR INJURY Pharmacia Corporation (US) 2006-06-21 EP disclosed
CN-1662490-A Nitrooxyderivatives of cyclooxygenase-2 inhibitors NICOX SA (FR) 2005-08-31 CN disclosed
WO-2005046615-A2 COMPOSITIONS FOR TREATMENT OF CENTRAL NERVOUS SYSTEM MEDIATED DISORDERS PHARMACIA & UPJOHN COMPANY LLC (US) 2005-05-26 WO disclosed
WO-2005037193-A2 COMPOSITIONS OF A CYCLOOXYGENASE-2 SELECTIVE INHIBITOR ADMINISTERED UNDER HYPOTHERMIC CONDITIONS FOR THE TREATMENT OF ISCHEMIC MEDIATED CENTRAL NERVOUS SYSTEM DISORDERS OR INJURY PHARMACIA CORPORATION (US) 2005-04-28 WO disclosed