SCHEMBL6025178

SCHEMBL6025178

N#CN1C=CCc2ccccc21

nearest known ligand 0.36

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.36
CA2 P00918 2/20 0.36
USP7 Q93009 1/20 0.32
ALDH1A1 P00352 2/20 0.31
GAA P10253 1/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
HPGD P15428 1/20 0.31
HTT P42858 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
HTR2A P28223 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9639131 0.87 CA1 (0.33) CA1CA2USP7ALDH1A1HPGD
SCHEMBL6615965 0.81 NPC1 (0.33) HPGDHTR2A
SCHEMBL3736107 0.74
SCHEMBL374979 0.71 ALDH1A1 (0.33) ALDH1A1MAPTHPGDHTR2A
SCHEMBL1198917 0.69 ALDH1A1 (0.36) ALDH1A1LMNAMAPTHPGDHTT
SCHEMBL15010759 0.69 POLB (0.33) ALDH1A1HPGDHTR2A
SCHEMBL4838387 0.69 HTR2A (0.36) ALDH1A1HPGDHTR2A
SCHEMBL2073990 0.69 HTR2A (0.36) ALDH1A1HPGDHTR2A
SCHEMBL1375450 0.69 NPC1 (0.35) ALDH1A1HPGDHTR2A
SCHEMBL553792 0.69 NPC1 (0.35) ALDH1A1HPGDHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1506178-A4 BICYCLIC MODULATORS OF ANDROGEN RECEPTOR FUNCTION BRISTOL MYERS SQUIBB CO (US) 2006-05-24 EP disclosed
EP-1506178-A2 BICYCLIC MODULATORS OF ANDROGEN RECEPTOR FUNCTION Bristol-Myers Squibb Company (US) 2005-02-16 EP disclosed
WO-2003096980-A2 BICYCLIC MODULATORS OF ANDROGEN RECEPTOR FUNCTION BRISTOL-MYERS SQUIBB COMPANY (US) 2003-11-27 WO disclosed