SCHEMBL6028341

SCHEMBL6028341

COc1c(-c2ccccc2)cc2c(c1C)NC(=O)CN=C2c1ccc(Br)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.47
TSHR P16473 1/20 0.47
ALOX12 P18054 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.46
ALDH1A1 P00352 1/20 0.45
GABRA1 P14867 3/20 0.44
GABRA5 P31644 3/20 0.44
GABRA3 P34903 3/20 0.44
GABRA2 P47869 3/20 0.44
GABRB2 P47870 3/20 0.44
GABRG2 P18507 2/20 0.44
GABRB3 P28472 2/20 0.44
TUBB4A P04350 2/20 0.44
TUBB P07437 2/20 0.44
TUBA3C P0DPH7 2/20 0.44
TUBA1B P68363 2/20 0.44
TUBA4A P68366 2/20 0.44
TUBB4B P68371 2/20 0.44
TUBB3 Q13509 2/20 0.44
TUBB2A Q13885 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6028351 0.91 KMT2A (0.54) MAPTTSHRALOX12ALDH1A1GABRA1
SCHEMBL5034663 0.79 KMT2A (0.54) MAPTTSHRALOX12SMN1; SMN2GABRA1
SCHEMBL4709491 0.78 TUBB4A (0.55) MAPTTSHRALOX12SMN1; SMN2ALDH1A1
SCHEMBL6028587 0.78 TUBB4A (0.51) ALDH1A1GABRA1GABRA5GABRA3GABRA2
SCHEMBL6268726 0.74 TUBB4A (0.53) TSHRALDH1A1GABRA1GABRA5GABRA3
SCHEMBL6669471 0.74 ALDH1A1 (0.53) MAPTTSHRALOX12SMN1; SMN2ALDH1A1
SCHEMBL18166499 0.74 GABRA1 (0.56) MAPTTSHRALOX12SMN1; SMN2ALDH1A1
SCHEMBL5490530 0.71 TUBB4A (0.55) SMN1; SMN2GABRA1GABRA5GABRA3GABRA2
SCHEMBL1365846 0.70 GABRA1 (0.69) MAPTTSHRALOX12SMN1; SMN2GABRA1
SCHEMBL1421181 0.70 KMT2A (0.82) MAPTTSHRALOX12ALDH1A1GABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1697332-A1 BENZO'1,4 ! DIAZEPIN-2-ONE DERIVATIVES AS PHOSPHODIESTERASE PDE2 INHIBITORS, PREPARATION AND THERAPEUTIC USE THEREOF NEURO3D (FR) 2006-09-06 EP disclosed
WO-2005063723-A1 BENZO`1,4 ! DIAZEPIN-2-ONE DERIVATIVES AS PHOSPHODIESTERASE PDE2 INHIBITORS, PREPARATION AND THERAPEUTIC USE THEREOF NEURO3D (FR) 2005-07-14 WO disclosed