SCHEMBL60299

SCHEMBL60299

C=C(C)N(C(=O)O)c1cc(C(F)(F)F)ccn1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.39
NOS2 P35228 1/20 0.39
ALDH1A1 P00352 3/20 0.38
GAA P10253 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
KDM4E B2RXH2 2/20 0.38
USP2 O75604 1/20 0.38
HPGD P15428 1/20 0.38
CYP2C19 P33261 1/20 0.38
HSD17B10 Q99714 1/20 0.38
POLQ O75417 1/20 0.37
KMO O15229 1/20 0.36
SORT1 Q99523 5/20 0.36
NR4A1 P22736 1/20 0.35
NR4A2 P43354 1/20 0.35
NR4A3 Q92570 1/20 0.35
ADRB2 P07550 1/20 0.35
MAPT P10636 1/20 0.34
SRD5A2 P31213 1/20 0.33
PROKR1 Q8TCW9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13570887 0.79 POLQ (0.45) NOS3NOS2ALDH1A1GAAL3MBTL1
SCHEMBL7985481 0.73 POLQ (0.41) NOS3NOS2ALDH1A1GAAL3MBTL1
SCHEMBL57464 0.72 POLQ (0.40) NOS3NOS2L3MBTL1HPGDHSD17B10
SCHEMBL1344896 0.71 NOS3 (0.52) NOS3NOS2ALDH1A1GAAL3MBTL1
SCHEMBL18137034 0.69 ADRB2 (0.39) NOS3NOS2ALDH1A1GAAL3MBTL1
SCHEMBL59042 0.69 PPARG (0.40) NOS3NOS2HPGDKMO
SCHEMBL15903091 0.69 GLA (0.41) GAAHPGDHSD17B10POLQADRB2
SCHEMBL29553421 0.68 NOS3 (0.48) NOS3NOS2ALDH1A1GAAL3MBTL1
SCHEMBL3216629 0.68 NOS3 (0.53) NOS3NOS2ALDH1A1GAAL3MBTL1
SCHEMBL8563867 0.68 NOS3 (0.48) NOS3NOS2ALDH1A1GAAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8143393-B2 Substituted 4-amino-pyrrolotriazine derivatives useful for treating hyper-proliferative disorders and diseases associated with angiogenesis BAYER HEALTHCARE LLC (US) 2012-03-27 US disclosed