SCHEMBL6030967

SCHEMBL6030967

Cn1ccc2cccc(CC(N)=O)c21

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CMA1 P23946 1/20 0.48
LMNA P02545 1/20 0.40
CDK4 P11802 4/20 0.36
CCND1 P24385 4/20 0.36
CCNE2 O96020 3/20 0.36
CCNE1 P24864 3/20 0.36
CDK2 P24941 3/20 0.36
PLA2G2A P14555 1/20 0.35
ICMT O60725 1/20 0.35
OXER1 Q8TDS5 1/20 0.35
PRKACA P17612 1/20 0.35
PRKACG P22612 1/20 0.35
PRKACB P22694 1/20 0.35
CAMK2B Q13554 1/20 0.35
CAMK2G Q13555 1/20 0.35
CAMK2D Q13557 1/20 0.35
CAMK2A Q9UQM7 1/20 0.35
GAA P10253 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11005480 0.79 CMA1 (0.48) CMA1CDK4CCND1CCNE2CCNE1
SCHEMBL28919591 0.79 CMA1 (0.44) CMA1SMN1; SMN2TDP1
SCHEMBL689243 0.78 CMA1 (0.47) CMA1CDK4CCND1CCNE2CCNE1
SCHEMBL3132206 0.78 CMA1 (0.44) CMA1CDK4CCND1CCNE2CCNE1
SCHEMBL3670913 0.76 CMA1 (0.60) CMA1CDK4CCND1CCNE2CCNE1
Hydrochloric Acid SCHEMBL26107888 0.76 CMA1 (0.43) CMA1CDK4CCND1CCNE2CCNE1
SCHEMBL2259757 0.75 ICMT (0.48) LMNAICMTGAANPSR1
SCHEMBL30006444 0.75 LGMN (0.38) ICMTHTT
SCHEMBL9275405 0.75 PARP1 (0.44) CMA1GAAADRA1DADRA1AADRA1B
SCHEMBL30082247 0.75 PARP1 (0.44) CMA1GAAADRA1DADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7109229-B2 Methods and compounds for treating proliferative diseases ELI LILLY AND COMPANY (US) 2006-09-19 US disclosed
EP-1325011-B1 METHODS AND COMPOUNDS FOR TREATING PROLIFERATIVE DISEASES LILLY CO ELI (US) 2004-05-06 EP disclosed
US-20040048915-A1 Methods and compounds for treating proliferative diseases ENGLER THOMAS ALBERT (US) 2004-03-11 US disclosed
EP-1325011-A2 METHODS AND COMPOUNDS FOR TREATING PROLIFERATIVE DISEASES ELI LILLY AND COMPANY (US) 2003-07-09 EP disclosed
WO-2002028861-A2 METHODS AND COMPOUNDS FOR TREATING PROLIFERATIVE DISEASES ELI LILLY AND COMPANY (US) 2002-04-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040048915-A1 Methods and compounds for treating proliferative diseases CDK4, CCNI, CCNA1 CMA1 2686/4885LMNA 1198/4885CDK4 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.