SCHEMBL6032032

SCHEMBL6032032

COc1c2c(c(C(=O)O)n(C)c1=O)CCN(Cc1cccc(Cl)c1F)C2=O

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 13/20 0.43
POLB P06746 1/20 0.35
LMNA P02545 1/20 0.35
HTR1D P28221 1/20 0.34
HTR1B P28222 1/20 0.34
CMA1 P23946 1/20 0.34
PCSK9 Q8NBP7 1/20 0.34
ALDH1A1 P00352 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4495597 0.83 AKR1B1 (0.43) P2RX7LMNAALDH1A1SMN1; SMN2
SCHEMBL4489713 0.82 CCR2 (0.38) P2RX7LMNASMN1; SMN2
SCHEMBL5449354 0.78 P2RX7 (0.38) P2RX7PCSK9
SCHEMBL4478430 0.75 LMNA (0.43) P2RX7POLBLMNAALDH1A1SMN1; SMN2
SCHEMBL4493255 0.74 MEN1 (0.46) POLBLMNAALDH1A1SMN1; SMN2
SCHEMBL4477879 0.74 MEN1 (0.38) P2RX7LMNAALDH1A1SMN1; SMN2
SCHEMBL4480439 0.73 P2RX7 (0.35) P2RX7SMN1; SMN2
SCHEMBL4482091 0.72 FSCN1 (0.34) P2RX7LMNAALDH1A1SMN1; SMN2
SCHEMBL4477812 0.72 LMNA (0.46) LMNAALDH1A1SMN1; SMN2
SCHEMBL4484366 0.71 CCR2 (0.39) P2RX7LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1725556-A1 HIV INTEGRASE INHIBITORS Merck & Co., Inc. (US) 2006-11-29 EP disclosed
WO-2005087768-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 2005-09-22 WO disclosed