SCHEMBL6032115

SCHEMBL6032115

O=C(O)Nc1cc(C(O)c2cc(F)ccc2F)c(Cl)cn1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 10/20 0.39
CES2 O00748 1/20 0.38
CES1 P23141 1/20 0.38
MAOB P27338 2/20 0.38
RAB9A P51151 4/20 0.38
NPC1 O15118 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
ALDH1A1 P00352 1/20 0.38
PKM P14618 1/20 0.38
TSHR P16473 1/20 0.38
LMNA P02545 1/20 0.37
KMT2A Q03164 1/20 0.37
FFAR2 O15552 1/20 0.36
KCNQ3 O43525 1/20 0.35
KCNQ2 O43526 1/20 0.35
KCNE1 P15382 1/20 0.35
KCNQ1 P51787 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12724232 0.83 CDK9 (0.44) ABL1
SCHEMBL1630845 0.79 CES2 (0.42) CES2CES1KCNQ3KCNQ2KCNE1
SCHEMBL6032853 0.79 KCNQ3 (0.38) ABL1MAOBRAB9ANPC1LMNA
SCHEMBL1633986 0.77 CES2 (0.37) CES2CES1
SCHEMBL1633909 0.77 CES2 (0.37) CES2CES1
SCHEMBL6032800 0.75 PSEN1 (0.49) MAOBRAB9ANPC1SMN1; SMN2ALDH1A1
SCHEMBL6032081 0.75 NPC1 (0.39) ABL1RAB9ANPC1SMN1; SMN2ALDH1A1
SCHEMBL6032111 0.74 PSEN1 (0.41) ALDH1A1PKMLMNA
SCHEMBL1632790 0.74 CES2 (0.34) CES2CES1KCNQ3KCNQ2KCNE1
SCHEMBL6032766 0.73 PSEN1 (0.49) ABL1RAB9ANPC1SMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1640366-A1 HETEROCYCLIC METHYL SULFONE DERIVATIVE DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2006-03-29 EP disclosed