SCHEMBL6032402

SCHEMBL6032402

N#Cc1ccc([CH]Cc2ccc(C#N)cc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 2/20 0.50
CYP2A6 P11509 2/20 0.50
IDO1 P14902 2/20 0.44
MAOB P27338 4/20 0.42
MAOA P21397 3/20 0.42
HTT P42858 1/20 0.42
GAA P10253 2/20 0.41
ALDH1A1 P00352 2/20 0.41
KCNJ1 P48048 1/20 0.41
KCNH2 Q12809 1/20 0.41
KDM4E B2RXH2 1/20 0.41
LMNA P02545 1/20 0.41
CYP19A1 P11511 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
FBP1 P09467 1/20 0.40
CA12 O43570 1/20 0.39
CA2 P00918 1/20 0.39
CA3 P07451 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7666461 0.91 CYP2A6 (0.68) LOXL2CYP2A6IDO1MAOBMAOA
SCHEMBL3410482 0.91 MAOA (0.56) LOXL2CYP2A6IDO1MAOBMAOA
SCHEMBL5208544 0.90 MAOB (0.53) LOXL2CYP2A6MAOBMAOAHTT
SCHEMBL4304998 0.88 NPC1 (0.44) LOXL2CYP2A6MAOBMAOAGAA
SCHEMBL6435082 0.88 NPC1 (0.44) LOXL2CYP2A6MAOBMAOAGAA
SCHEMBL10804609 0.86 MAOB (0.44) LOXL2CYP2A6IDO1MAOBMAOA
SCHEMBL19437177 0.82 MAOB (0.41) LOXL2CYP2A6IDO1MAOBMAOA
SCHEMBL10671045 0.79 LOXL2 (0.47) LOXL2CYP2A6IDO1MAOBMAOA
SCHEMBL10671048 0.79 LOXL2 (0.47) LOXL2CYP2A6IDO1MAOBMAOA
SCHEMBL17855518 0.79 LOXL2 (0.47) LOXL2CYP2A6IDO1MAOBMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1661886-A1 INSECTICIDE FOR AGRICULTURAL OR HORTICULTURAL USE AND METHOD OF USE THEREOF Mitsui Chemicals, Inc. (JP) 2006-05-31 EP disclosed
US-5811422-A USEFUL FOR TREATING VIRAL INFECTIONS THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1998-09-22 US disclosed
US-5610294-A VIRAL TREATMENT THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1997-03-11 US disclosed