SCHEMBL6036281

SCHEMBL6036281

CC(C)(C)OC(=O)CC[C@H](NC(=O)Oc1ccc(C=O)cc1)C(=O)OC(C)(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.43
PPARG P37231 5/20 0.36
PPARA Q07869 5/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
HTT P42858 1/20 0.36
APP P05067 1/20 0.35
ADRB2 P07550 1/20 0.35
ADRB1 P08588 1/20 0.35
ADRB3 P13945 1/20 0.35
ELANE P08246 1/20 0.35
TDP1 Q9NUW8 1/20 0.34
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
PPARD Q03181 2/20 0.34
ACHE P22303 1/20 0.34
KDM4E B2RXH2 1/20 0.33
NPC1 O15118 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6036278 1.00 KMT2A (0.43) KMT2APPARGPPARACYP1A2CYP2C9
SCHEMBL6036686 0.83 PPARA (0.40) PPARGPPARATDP1PPARDKDM4E
SCHEMBL6036690 0.83 PPARA (0.40) PPARGPPARATDP1PPARDKDM4E
SCHEMBL29170202 0.82 PPARG (0.48) KMT2APPARGPPARACYP1A2ACHE
SCHEMBL7903853 0.82 PPARG (0.48) KMT2APPARGPPARACYP1A2ACHE
SCHEMBL7902134 0.81 PPARG (0.34) KMT2APPARGPPARAELANETDP1
SCHEMBL7903878 0.80 PPARG (0.34) PPARGPPARACYP1A2CYP2C9CYP2C19
SCHEMBL7894784 0.80 PPARG (0.34) PPARGPPARAELANETDP1NFKB1
SCHEMBL13570965 0.77 CYP1A2 (0.50) KMT2APPARGPPARACYP1A2CYP2C9
SCHEMBL13570964 0.77 CYP1A2 (0.50) KMT2APPARGPPARACYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1644025-A4 WATER-SOLUBLE SHPS AS NOVEL ALKYLATING AGENTS VION PHARMACEUTICALS INC (US) 2006-11-15 EP disclosed
EP-1644025-A1 WATER-SOLUBLE SHPS AS NOVEL ALKYLATING AGENTS Vion Pharmaceuticals, Inc. (US) 2006-04-12 EP disclosed
US-20050043244-A1 Water-soluble SHPs as novel alkylating agents VION PHARMACEUTICALS, INC. (US) 2005-02-24 US disclosed
US-6855695-B2 Water-soluble SHPs as novel alkylating agents VION PHARMACEUTICALS, INC. (US) 2005-02-15 US disclosed
WO-2005004897-A1 WATER-SOLUBLE SHPS AS NOVEL ALKYLATING AGENTS VION PHARMACEUTICALS, INC. (US) 2005-01-20 WO disclosed
US-20040254103-A1 WATER-SOLUBLE SHPS AS NOVEL ALKYLATING AGENTS NANOSHIFT, LLC 2004-12-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040254103-A1 WATER-SOLUBLE SHPS AS NOVEL ALKYLATING AGENTS SHPRH, OGFR, COG3 KMT2A 1653/4885PPARG 3545/4885PPARA 4021/4885
US-20050043244-A1 Water-soluble SHPs as novel alkylating agents GRM3, GRIA3, SHPRH KMT2A 2306/4885PPARG 2900/4885PPARA 3768/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.