SCHEMBL6038491

SCHEMBL6038491

O=C(O)N(C(=O)Oc1ccccc1)c1cc(Cl)ccn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 4/20 0.41
ATM Q13315 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
LIPE Q05469 2/20 0.39
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
ALDH1A1 P00352 3/20 0.37
MAPT P10636 2/20 0.37
LMNA P02545 3/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
PTGES O14684 1/20 0.36
KCNH2 Q12809 1/20 0.36
KDM4C Q9H3R0 1/20 0.36
KDM4E B2RXH2 3/20 0.35
USP2 O75604 1/20 0.35
ALOX15 P16050 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
OGT O15294 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5104290 0.94 L3MBTL1 (0.42) L3MBTL1ATMTDP1LIPECYP1A2
SCHEMBL5104294 0.82 L3MBTL1 (0.42) L3MBTL1TDP1ALDH1A1MAPTLMNA
SCHEMBL28753070 0.78 L3MBTL1 (0.45) L3MBTL1ATMTDP1LIPEALDH1A1
SCHEMBL5700035 0.72 MAPT (0.48) L3MBTL1TDP1ALDH1A1MAPTSMN1; SMN2
SCHEMBL12280370 0.71 CYP1A2 (0.36) L3MBTL1ATMTDP1LIPECYP1A2
SCHEMBL11076613 0.71 L3MBTL1 (0.53) L3MBTL1ATMTDP1LIPEALDH1A1
SCHEMBL3556176 0.71 MAOA (0.45) L3MBTL1ATMTDP1CYP3A4ALDH1A1
SCHEMBL12420813 0.71 L3MBTL1 (0.45) L3MBTL1ATMTDP1LIPEALDH1A1
SCHEMBL6687991 0.70 L3MBTL1 (0.66) L3MBTL1ATMTDP1LIPEALDH1A1
SCHEMBL27745477 0.69 MAPT (0.45) L3MBTL1CYP1A2CYP3A4CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116903526-A Pyridinylpyridinone compounds 思普瑞特生物科学公司 2023-10-20 CN disclosed
CN-116891431-A Pyridinylpyridinone compounds 思普瑞特生物科学公司 2023-10-17 CN disclosed
CN-111094244-B Pyridinylpyridinone compounds 思普瑞特生物科学公司 2023-07-11 CN disclosed
US-20060004029-A1 Nitrogen-containing aromatic derivatives EISAI R&D MANAGEMENT CO., LTD. (JP) 2006-01-05 US disclosed
EP-1522540-A1 AZAARENE DERIVATIVES Eisai Co., Ltd. (JP) 2005-04-13 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060004029-A1 Nitrogen-containing aromatic derivatives NR0B2, NR0B1, NR4A1 L3MBTL1 2633/4885ATM 2354/4885TDP1 4358/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.