SCHEMBL604040

SCHEMBL604040

O=C(O)[C@H](Br)c1ccccc1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 3/20 0.76
CES1 P23141 3/20 0.76
SRC P12931 2/20 0.59
CYP2D6 P10635 1/20 0.59
LMNA P02545 3/20 0.56
MAPK1 P28482 1/20 0.56
TDP1 Q9NUW8 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
HDAC3 O15379 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC10 Q969S8 1/20 0.44
HDAC11 Q96DB2 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
HDAC9 Q9UKV0 1/20 0.44
HDAC5 Q9UQL6 1/20 0.44
CYP1A2 P05177 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzene SCHEMBL28201061 1.00 CES2 (0.76) CES2CES1SRCCYP2D6LMNA
SCHEMBL234580 1.00 CES2 (0.76) CES2CES1SRCCYP2D6LMNA
SCHEMBL5899350 1.00 CES2 (0.76) CES2CES1SRCCYP2D6LMNA
Ammonia Solution, Strong SCHEMBL38660268 0.97 CES2 (0.73) CES2CES1SRCCYP2D6LMNA
Hydrochloric Acid SCHEMBL7037834 0.97 CES2 (0.73) CES2CES1SRCCYP2D6LMNA
Methane SCHEMBL6115781 0.97 CES2 (0.73) CES2CES1SRCCYP2D6LMNA
Alcohol SCHEMBL29064519 0.89 CES2 (0.61) CES2CES1SRCCYP2D6LMNA
SCHEMBL5820145 0.86 CES2 (0.73) CES2CES1SRCCYP2D6LMNA
SCHEMBL7437238 0.85 PTGS2 (0.61) CES2CES1SRCCYP2D6CYP1A2
SCHEMBL4973413 0.84 CES2 (0.77) CES2CES1SRCCYP2D6LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 26 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120041225-A1 KIT FOR AUTOMATED RESOLVING AGENT SELECTION AND METHOD THEREOF VAIDYA NITEEN A (US) 2012-02-16 US claimed
EP-1981831-A2 KIT FOR AUTOMATED RESOLVING AGENT SELECTION AND METHOD THEREOF Vaidya, Niteen A. (US) 2008-10-22 EP claimed
WO-2007092264-A2 KIT FOR AUTOMATED RESOLVING AGENT SELECTION AND METHOD THEREOF VAIDYA NITEEN A (US) 2007-08-16 WO claimed
US-20070185346-A1 Kit for automated resolving agent selection and method thereof VAIDYA NITEEN A 2007-08-09 US claimed
US-20120041225-A1 KIT FOR AUTOMATED RESOLVING AGENT SELECTION AND METHOD THEREOF VAIDYA NITEEN A (US) 2012-02-16 US disclosed
EP-1981831-A2 KIT FOR AUTOMATED RESOLVING AGENT SELECTION AND METHOD THEREOF Vaidya, Niteen A. (US) 2008-10-22 EP disclosed
WO-2007126258-A1 THE METHOD OF MAKING OPTICALLY ACTIVE 2-HALO-2-(N-SUBSTITUTED PHENYL)ACETIC ACID ESTERS AND 2-HALO-2-(N-SUBSTITUTED PHENYL)ACETIC ACIDS BY ENZYMATIC METHOD ENZYTECH, LTD (KR) 2007-11-08 WO disclosed
WO-2007092264-A2 KIT FOR AUTOMATED RESOLVING AGENT SELECTION AND METHOD THEREOF VAIDYA NITEEN A (US) 2007-08-16 WO disclosed
US-20070185346-A1 Kit for automated resolving agent selection and method thereof VAIDYA NITEEN A 2007-08-09 US disclosed
US-7084140-B2 Arylglycinamide derivatives, method of producing said derivatives and pharmaceutical compositions containing these compounds BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2006-08-01 US disclosed
US-20030092704-A1 Novel arylglycinamide derivatives, method of producing said derivatives and pharmaceutical compositions containing these compounds BOEHRINGER INGELHEIM PHARMA KG (DE) 2003-05-15 US disclosed
US-6498162-B1 TREATING INFLAMMATORY AND ALLERGIC DISEASES OF RESPIRATORY TRACT AND DISEASES OF CENTRAL NERVOUS SYSTEM BOEHRINGER INGELHEIM PHARMA KG (DE) 2002-12-24 US disclosed
US-6251909-B1 Arylglycinamide derivatives, methods of producing these substances and pharmaceutical compositions containing such compounds BOEHRINGER INGELHEIM KG (DE) 2001-06-26 US disclosed
US-6124296-A NEUROKININ (TACHYKININ) ANTAGONISTS BOEHRINGER INGELHEIM KG (DE) 2000-09-26 US disclosed
US-5801274-A N- mercaptoacyl(amino acid or peptide)! compounds and S-lipophilic aliphatic carbonyl derivatives thereof as antihypertensives INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (FR) 1998-09-01 US disclosed
US-5591891-A PEPTIDASE INHIBITORS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 1997-01-07 US disclosed
WO-1994017036-A1 S-LIPOPHILIC ALIPHATIC CARBONYL [N-MERCAPTOACYL-(AMINO ACID OR PEPTIDE)] COMPOUNDS AS ANTIHYPERTENSIVE AGENTS INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 1994-08-04 WO disclosed
EP-0595878-A1 ACYLMERCAPTOALKANOYLDIPEPTIDES, METHODS OF PREPARATION AND THEIR THERAPEUTIC USE INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 1994-05-11 EP disclosed
WO-1993002099-A1 ACYLMERCAPTOALKANOYLDIPEPTIDES, METHODS OF PREPARATION AND THEIR THERAPEUTIC USE INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 1993-02-04 WO disclosed
EP-0524553-A1 Acylmercaptoalkanoyldipeptides, methods of preparation and their therapeutic use INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM) (FR) 1993-01-27 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120041225-A1 KIT FOR AUTOMATED RESOLVING AGENT SELECTION AND METHOD THEREOF ACKR3, KIT, C3AR1 CES2 1677/4885CES1 213/4885SRC 4485/4885
US-20030092704-A1 Novel arylglycinamide derivatives, method of producing said derivatives and pharmaceutical compositions containing these compounds GCGR, NGLY1, CCKAR CES2 1591/4885CES1 1684/4885SRC 2832/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.