SCHEMBL6047610

SCHEMBL6047610

COc1ccc(C2=C(Cl)C(Cl)=CC[CH]2)c(-c2cccc(F)c2F)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
AMY1A P0DUB6 3/20 0.34
CYP11B1 P15538 3/20 0.33
CYP11B2 P19099 3/20 0.33
PDE2A O00408 1/20 0.32
PDE10A Q9Y233 1/20 0.32
MAPK14 Q16539 2/20 0.31
KDM4E B2RXH2 2/20 0.31
ALDH1A1 P00352 2/20 0.31
GAA P10253 2/20 0.31
MAPT P10636 2/20 0.31
FLT3 P36888 1/20 0.31
ALOX15 P16050 1/20 0.31
TSHR P16473 1/20 0.31
MAPK1 P28482 1/20 0.31
HSD17B10 Q99714 1/20 0.31
CYP17A1 P05093 2/20 0.31
PTGES O14684 1/20 0.31
DYRK3 O43781 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6047654 0.83 NUDT1 (0.42) NPC1RAB9ACYP11B1CYP11B2MAPK14
SCHEMBL6047650 0.81 CYP24A1 (0.40) NPC1RAB9AMAPK14KDM4EALDH1A1
SCHEMBL6047634 0.79 CYP1A1 (0.40) PDE2AMAPK14CYP1A1CYP1A2CYP2E1
SCHEMBL6047612 0.78 MAOB (0.40) RAB9AMAPK14KDM4EALDH1A1GAA
SCHEMBL6047630 0.77 CYP3A4 (0.39) CYP11B1CYP11B2MAPK14ALDH1A1CYP17A1
SCHEMBL6047641 0.76 ALKBH3 (0.34) RAB9ACYP11B1CYP11B2ALDH1A1GAA
SCHEMBL6047586 0.74 CHRNA7 (0.35) NPC1RAB9AKDM4EMAPTALOX15
SCHEMBL18436302 0.72 CD274 (0.48) NPC1RAB9AAMY1ACYP11B1CYP11B2
SCHEMBL6047626 0.72 NPC1 (0.36) NPC1RAB9APDE2APDE10AKDM4E
SCHEMBL29048448 0.64 RAB9A (0.51) NPC1RAB9AAMY1AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2006501194-A 2006-01-12 JP claimed
EP-1525190-A1 CCK-1 RECEPTOR MODULATORS JANSSEN PHARMACEUTICA N.V. (BE) 2005-04-27 EP claimed
WO-2004007463-A1 CCK-1 RECEPTOR MODULATORS JANSSEN PHARMACEUTICA, N.V. (BE) 2004-01-22 WO claimed