SCHEMBL6047633

SCHEMBL6047633

COc1ccc(C2=CC(Oc3ccccc3)=CC[CH]2)c(-c2cc(C)cc(C)c2)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.36
LTA4H P09960 1/20 0.36
IDH1 O75874 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
NAAA Q02083 2/20 0.33
KDM4E B2RXH2 2/20 0.33
HDAC8 Q9BY41 1/20 0.33
MAPT P10636 1/20 0.33
MAPK1 P28482 1/20 0.33
GRIN1 Q05586 1/20 0.32
GRIN2B Q13224 1/20 0.32
MAOB P27338 1/20 0.32
ACHE P22303 2/20 0.32
BACE1 P56817 1/20 0.32
CYP19A1 P11511 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
GAA P10253 1/20 0.32
CYP2C9 P11712 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6047600 0.91 ACHE (0.39) PTPN1LTA4HSMN1; SMN2NAAAKDM4E
SCHEMBL6047648 0.88 NAAA (0.42) PTPN1LTA4HNAAACYP1A2CYP3A4
SCHEMBL6047602 0.83 NAAA (0.37) PTPN1LTA4HSMN1; SMN2NAAAKDM4E
SCHEMBL6047613 0.83 THRA (0.39) PTPN1SMN1; SMN2NAAAKDM4EMAPT
SCHEMBL6047656 0.82 HCRTR1 (0.36) PTPN1NAAAHDAC8GRIN2BL3MBTL1
SCHEMBL6047594 0.81 NAAA (0.40) PTPN1LTA4HSMN1; SMN2NAAAKDM4E
SCHEMBL6047659 0.81 THRA (0.39) PTPN1NAAABACE1
SCHEMBL6047596 0.80 ABL1 (0.45) PTPN1LTA4HSMN1; SMN2NAAAKDM4E
SCHEMBL6047642 0.80 MAOB (0.42) PTPN1KDM4EHDAC8MAPTMAOB
SCHEMBL6047590 0.79 MEN1 (0.41) SMN1; SMN2MAPTMAOBALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2006501194-A 2006-01-12 JP claimed
EP-1525190-A1 CCK-1 RECEPTOR MODULATORS JANSSEN PHARMACEUTICA N.V. (BE) 2005-04-27 EP claimed
WO-2004007463-A1 CCK-1 RECEPTOR MODULATORS JANSSEN PHARMACEUTICA, N.V. (BE) 2004-01-22 WO claimed