SCHEMBL6047646

SCHEMBL6047646

COC1=CC[CH]C(c2c(Cl)cccc2Cl)=C1c1ccc(C)cc1

nearest known ligand 0.32

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
HPGD P15428 1/20 0.32
ALOX15 P16050 1/20 0.32
CYP2C19 P33261 1/20 0.32
HSD17B10 Q99714 1/20 0.32
ALKBH3 Q96Q83 1/20 0.30
GRIA1 P42261 1/20 0.30
CACNG8 Q8WXS5 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6047579 0.90 GRIA1 (0.31) GRIA1CACNG8
SCHEMBL5887426 0.85 MEN1 (0.34) CYP2D6CYP2C9HPGDALOX15CYP2C19
SCHEMBL5887320 0.82 ACHE (0.33) CYP2D6CYP2C9HPGDALOX15CYP2C19
SCHEMBL5887143 0.82 PTGS2 (0.35) CYP2D6CYP2C9HPGDALOX15CYP2C19
SCHEMBL5887105 0.82 ESR2 (0.35)
SCHEMBL6047593 0.81 ALKBH3 (0.36) CYP2D6CYP2C9HPGDALOX15CYP2C19
SCHEMBL5887353 0.80 MEN1 (0.35) HSD17B10ALKBH3
SCHEMBL5887285 0.77 ALKBH3 (0.44) CYP2C9HPGDCYP2C19HSD17B10ALKBH3
SCHEMBL5887287 0.77 ACHE (0.46) HPGDALKBH3
SCHEMBL5887347 0.77 MEN1 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2006501194-A 2006-01-12 JP claimed
EP-1525190-A1 CCK-1 RECEPTOR MODULATORS JANSSEN PHARMACEUTICA N.V. (BE) 2005-04-27 EP claimed
WO-2004007463-A1 CCK-1 RECEPTOR MODULATORS JANSSEN PHARMACEUTICA, N.V. (BE) 2004-01-22 WO claimed