SCHEMBL6058797

SCHEMBL6058797

C=Cc1cc(CC(C(=O)OCC)C(=O)OCC)cnc1NC(=O)OC(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 3/20 0.36
SMN1; SMN2 Q16637 3/20 0.34
PKM P14618 1/20 0.34
MKNK2 Q9HBH9 1/20 0.34
ALDH1A1 P00352 2/20 0.33
TP53 P04637 1/20 0.33
MMP8 P22894 1/20 0.33
L3MBTL1 Q9Y468 2/20 0.32
AAK1 Q2M2I8 1/20 0.32
MAPK1 P28482 1/20 0.32
IRAK4 Q9NWZ3 1/20 0.32
LCK P06239 1/20 0.32
MAP4K4 O95819 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
HTT P42858 1/20 0.31
PPARA Q07869 1/20 0.31
CPB2 Q96IY4 1/20 0.31
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Malonic Acid Diethyl Ester SCHEMBL7380431 0.96 PPARG (0.36) PPARGSMN1; SMN2PKMMKNK2ALDH1A1
SCHEMBL6058628 0.96 PPARG (0.39) PPARGSMN1; SMN2PKMMKNK2ALDH1A1
SCHEMBL6059446 0.86 CPB2 (0.41) PPARGSMN1; SMN2PKMMKNK2ALDH1A1
SCHEMBL6059053 0.85 SMN1; SMN2 (0.36) PPARGSMN1; SMN2PKMMKNK2ALDH1A1
SCHEMBL6058805 0.84 PPARG (0.34) PPARGMAPK1PPARA
SCHEMBL6059174 0.82 PPARG (0.34) PPARGMKNK2AAK1LCKMAP4K4
Malonic Acid Diethyl Ester SCHEMBL7380709 0.82 L3MBTL1 (0.41) PPARGPKMMKNK2ALDH1A1L3MBTL1
SCHEMBL6059338 0.82 LCK (0.40) AAK1MAPK1LCKMAP4K4
SCHEMBL6060000 0.82 CPB2 (0.39) PPARGPKMMKNK2ALDH1A1TP53
SCHEMBL6059191 0.81 MAP4K4 (0.35) AAK1MAPK1LCKMAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7071175-B1 Pyridine mercapto carboxylic acids as carboxypeptidase U inhibitors ASTRAZENECA AB (SE) 2006-07-04 US disclosed
EP-1180098-A1 NEW COMPOUNDS AstraZeneca AB (SE) 2002-02-20 EP disclosed
WO-2000066557-A1 NEW COMPOUNDS ASTRAZENECA AB (SE) 2000-11-09 WO disclosed