SCHEMBL6060299

SCHEMBL6060299

CCCCOC(=O)c1ncc2ccccc2c1-c1ccc(C)cc1OCc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.43
CYP3A4 P08684 2/20 0.43
TSHR P16473 2/20 0.43
TDP1 Q9NUW8 2/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
MAPK1 P28482 1/20 0.43
PTGER1 P34995 4/20 0.39
PTGER4 P35408 1/20 0.39
PTGER3 P43115 1/20 0.39
PTGER2 P43116 1/20 0.39
GABRA1 P14867 4/20 0.39
GABRG2 P18507 4/20 0.39
GABRB3 P28472 4/20 0.39
GABRA5 P31644 4/20 0.39
GABRA3 P34903 4/20 0.39
GABRA2 P47869 4/20 0.39
MRGPRX4 Q96LA9 1/20 0.39
MAPT P10636 2/20 0.39
HPGD P15428 2/20 0.39
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6061077 0.86 KDM4E (0.43) ALDH1A1CYP3A4TSHRTDP1L3MBTL1
SCHEMBL27913218 0.77 TSHR (0.54) ALDH1A1CYP3A4TSHRTDP1L3MBTL1
SCHEMBL27653607 0.72 TSHR (0.50) ALDH1A1CYP3A4TSHRTDP1L3MBTL1
SCHEMBL6061205 0.72 TSHR (0.46) ALDH1A1CYP3A4TSHRTDP1L3MBTL1
SCHEMBL522404 0.71 L3MBTL1 (0.47) ALDH1A1CYP3A4TSHRTDP1L3MBTL1
SCHEMBL27404312 0.71 TSHR (0.52) ALDH1A1CYP3A4TSHRTDP1L3MBTL1
SCHEMBL6060652 0.69 TSHR (0.47) ALDH1A1CYP3A4TSHRTDP1L3MBTL1
SCHEMBL523256 0.69 TSHR (0.52) ALDH1A1CYP3A4TSHRTDP1L3MBTL1
SCHEMBL2805603 0.69 ALDH1A1 (0.61) ALDH1A1CYP3A4TSHRTDP1L3MBTL1
SCHEMBL8881493 0.68 TSHR (0.48) ALDH1A1CYP3A4TSHRTDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1644336-A1 NITROGEN-CONTAINING HETEROARYL COMPOUNDS AND THEIR USE IN INCREASING ENDOGENEOUS ERYTHROPOIETIN FIBROGEN, INC. (US) 2006-04-12 EP disclosed
WO-2004108681-A1 NITROGEN-CONTAINING HETEROARYL COMPOUNDS AND THEIR USE IN INCREASING ENDOGENOUS ERYTHROPOIETIN FIBROGEN, INC. (US) 2004-12-16 WO disclosed