SCHEMBL6061073

SCHEMBL6061073

CCOC(=O)CN1C(=O)c2ccc3ccccc3c2C1=O

nearest known ligand 0.62

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 1/20 0.62
PIN4 Q9Y237 1/20 0.62
ALDH1A1 P00352 4/20 0.52
MAPT P10636 1/20 0.48
HTT P42858 1/20 0.48
HSD17B10 Q99714 1/20 0.48
PTGS2 P35354 1/20 0.47
CASP3 P42574 1/20 0.47
GSK3A P49840 1/20 0.46
GSK3B P49841 1/20 0.46
NPSR1 Q6W5P4 1/20 0.45
CYP1A2 P05177 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
KMT2A Q03164 1/20 0.44
TNF P01375 1/20 0.44
KDM4E B2RXH2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1757427 0.85 CASP3 (0.44) PIN1PIN4ALDH1A1MAPTHSD17B10
SCHEMBL7549529 0.81 CA12 (0.60) ALDH1A1MAPTHSD17B10CYP1A2KMT2A
SCHEMBL523639 0.81 PIN1 (0.68) PIN1PIN4ALDH1A1MAPTHTT
SCHEMBL5998379 0.81 PIN1 (0.41) PIN1PIN4ALDH1A1CASP3KMT2A
SCHEMBL11453331 0.80 ALDH1A1 (0.77) PIN1PIN4ALDH1A1MAPTHTT
SCHEMBL18485415 0.80 KDM4E (0.45) ALDH1A1MAPTHSD17B10KMT2ATNF
SCHEMBL12235635 0.79 CYP1B1 (0.53) ALDH1A1MAPTHSD17B10NPSR1CYP1A2
SCHEMBL442751 0.77 PIN1 (1.00) PIN1PIN4ALDH1A1MAPTHTT
SCHEMBL11395567 0.77 PIN1 (0.75) PIN1PIN4ALDH1A1MAPTHTT
SCHEMBL25175089 0.76 PIN1 (0.61) PIN1PIN4ALDH1A1MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1644336-A1 NITROGEN-CONTAINING HETEROARYL COMPOUNDS AND THEIR USE IN INCREASING ENDOGENEOUS ERYTHROPOIETIN FIBROGEN, INC. (US) 2006-04-12 EP disclosed
WO-2004108681-A1 NITROGEN-CONTAINING HETEROARYL COMPOUNDS AND THEIR USE IN INCREASING ENDOGENOUS ERYTHROPOIETIN FIBROGEN, INC. (US) 2004-12-16 WO disclosed