Methaniazide

Methaniazide

SCHEMBL606355

O=C(NNCS(=O)(=O)O)c1ccncc1

nearest known ligand 0.66

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.60
HPGD P15428 2/20 0.55
HDAC3 O15379 1/20 0.55
HDAC1 Q13547 1/20 0.55
HDAC2 Q92769 1/20 0.55
KDM4E B2RXH2 1/20 0.52
MPO P05164 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
ADORA3 P0DMS8 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2A6 P11509 1/20 0.52
CYP2C19 P33261 1/20 0.52
TP53 P04637 1/20 0.51
GAA P10253 6/20 0.50
CA1 P00915 2/20 0.49
CA9 Q16790 2/20 0.49
MAOA P21397 1/20 0.49
MAOB P27338 1/20 0.49
PTGS2 P35354 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6926470 0.83 HDAC3 (0.60) ALDH1A1HPGDHDAC3HDAC1HDAC2
Methaniazide SCHEMBL29414958 0.82 ALDH1A1 (0.55) ALDH1A1HPGDHDAC3HDAC1HDAC2
Metazide SCHEMBL2109857 0.80 ALDH1A1 (0.72) ALDH1A1HPGDHDAC3HDAC1HDAC2
SCHEMBL2992964 0.77 ALDH1A1 (1.00) ALDH1A1HPGDKDM4EMPOCYP1A2
SCHEMBL2992165 0.77 ALDH1A1 (0.67) ALDH1A1HPGDKDM4EMPOCYP1A2
SCHEMBL2992612 0.77 HDAC3 (0.70) ALDH1A1HPGDHDAC3HDAC1HDAC2
SCHEMBL2998085 0.75 ALDH1A1 (0.64) ALDH1A1HPGDHDAC3HDAC1HDAC2
SCHEMBL2998521 0.75 HDAC3 (0.68) ALDH1A1HPGDHDAC3HDAC1HDAC2
SCHEMBL3001447 0.74 HDAC3 (0.81) ALDH1A1HDAC3HDAC1HDAC2KDM4E
SCHEMBL14113829 0.74 ALDH1A1 (0.62) ALDH1A1HPGDHDAC3HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 158 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3880688-B1 OLIGOSACCHARIDE PREPARATIONS AND COMPOSITIONS DSM IP ASSETS BV (NL) 2025-09-17 EP claimed
US-11655267-B2 Oligosaccharide preparations and compositions DSM IP ASSETS B.V. (NL) 2023-05-23 US claimed
US-20210395284-A1 OLIGOSACCHARIDE PREPARATIONS AND COMPOSITIONS DSM IP ASSETS B.V. (NL) 2021-12-23 US claimed
EP-3880688-A1 OLIGOSACCHARIDE PREPARATIONS AND COMPOSITIONS Midori USA, Inc. (US) 2021-09-22 EP claimed
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
US-20100226943-A1 SURFACE TOPOGRAPHIES FOR NON-TOXIC BIOADHESION CONTROL UNIVERSITY OF FLORIDA (US) 2010-09-09 US claimed
EP-1954244-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY Scidose, Llc (US) 2008-08-13 EP claimed
WO-2007061529-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY SCIDOSE LLC. (US) 2007-05-31 WO claimed
US-20070116729-A1 Lyophilization process and products obtained thereby SCIDOSE LLC 2007-05-24 US claimed
EP-1225916-A1 COMPOSITIONS AND METHODS FOR CONTROLLED-RELEASE DELIVERY AND INCREASED POTENCY OF PHARMACEUTICALS VIA HYDROPHOBIC ION-PAIRING University Technology Corporation (US) 2002-07-31 EP claimed
WO-2001032218-A1 COMPOSITIONS AND METHODS FOR CONTROLLED-RELEASE DELIVERY AND INCREASED POTENCY OF PHARMACEUTICALS VIA HYDROPHOBIC ION-PAIRING UNIVERSITY TECHNOLOGY CORPORATION (US) 2001-05-10 WO claimed
US-5596095-A REMOVAL OF NEOPENTYL PROTECTING GROUPS AND REGENERATION OF PARENT DRUGS PROCEPT, INC. (US) 1997-01-21 US claimed
EP-4687916-A1 OLIGOSACCHARIDE PREPARATION COUNTERACTING RESPIRATORY DISEASE EFFECT DSM IP Assets B.V. (NL) 2026-02-11 EP disclosed
EP-3880688-B1 OLIGOSACCHARIDE PREPARATIONS AND COMPOSITIONS DSM IP ASSETS BV (NL) 2025-09-17 EP disclosed
EP-4613755-A1 OLIGOSACCHARIDE PREPARATIONS AND COMPOSITIONS DSM IP Assets B.V. (NL) 2025-09-10 EP disclosed
US-12383570-B2 Methods of selectively modulating gastrointestinal microbial growth DSM IP ASSETS B.V. (NL) 2025-08-12 US disclosed
WO-1996040156-A1 DIPHOSPHONATE DERIVATIVES OF THERAPEUTIC AGENTS ELIZANOR BIOPHARMACEUTICALS, INC. (US) 1996-12-19 WO disclosed
EP-0741570-A1 METHOD FOR PREVENTING OR REDUCING PHOTOSENSITIVITY AND/OR PHOTOTOXICITY REACTIONS TO MEDICATIONS G.D. SEARLE & CO. (US) 1996-11-13 EP disclosed
WO-1996018609-A1 FORMATION AND UTILITY OF SULFONIC ACID PROTECTING GROUPS PROCEPT, INC. (US) 1996-06-20 WO disclosed
WO-1995020387-A1 METHOD FOR PREVENTING OR REDUCING PHOTOSENSITIVITY AND/OR PHOTOTOXICITY REACTIONS TO MEDICATIONS G.D. SEARLE & CO. (US) 1995-08-03 WO disclosed