SCHEMBL6926470

SCHEMBL6926470

O=C(NNCCS(=O)(=O)O)c1ccncc1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.60
HDAC1 Q13547 1/20 0.60
HDAC2 Q92769 1/20 0.60
ALDH1A1 P00352 1/20 0.56
HPGD P15428 2/20 0.53
CYP1A2 P05177 2/20 0.49
CYP2C19 P33261 2/20 0.49
TP53 P04637 1/20 0.49
KDM4E B2RXH2 1/20 0.49
MPO P05164 1/20 0.49
CYP3A4 P08684 1/20 0.49
ADORA3 P0DMS8 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2A6 P11509 1/20 0.49
GAA P10253 6/20 0.48
CA1 P00915 2/20 0.46
CA9 Q16790 2/20 0.46
MAOA P21397 1/20 0.46
MAOB P27338 1/20 0.46
PTGS2 P35354 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Methaniazide SCHEMBL606355 0.83 ALDH1A1 (0.60) HDAC3HDAC1HDAC2ALDH1A1HPGD
SCHEMBL2998521 0.80 HDAC3 (0.68) HDAC3HDAC1HDAC2ALDH1A1HPGD
SCHEMBL3001447 0.78 HDAC3 (0.81) HDAC3HDAC1HDAC2ALDH1A1CYP1A2
SCHEMBL2990093 0.77 HDAC3 (0.91) HDAC3HDAC1HDAC2ALDH1A1GAA
Metazide SCHEMBL2109857 0.77 ALDH1A1 (0.72) HDAC3HDAC1HDAC2ALDH1A1HPGD
SCHEMBL7401272 0.77 HDAC3 (0.64) HDAC3HDAC1HDAC2ALDH1A1CYP1A2
SCHEMBL2998122 0.76 HDAC3 (0.88) HDAC3HDAC1HDAC2GAANAAA
SCHEMBL17141675 0.75 HDAC3 (1.00) HDAC3HDAC1HDAC2ALDH1A1GAA
SCHEMBL2992964 0.74 ALDH1A1 (1.00) ALDH1A1HPGDCYP1A2CYP2C19TP53
SCHEMBL2992165 0.74 ALDH1A1 (0.67) ALDH1A1HPGDCYP1A2CYP2C19TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051655-A4 METHODS AND APPARATUS FOR ACCELERATED ORTHOKERATOLOGY ISTA PHARMACEUTICALS INC (US) 2003-03-19 EP disclosed
EP-1051655-A1 METHODS AND APPARATUS FOR ACCELERATED ORTHOKERATOLOGY Ista Pharmaceuticals, Inc. (US) 2000-11-15 EP disclosed
WO-1999039238-A1 METHODS AND APPARATUS FOR ACCELERATED ORTHOKERATOLOGY KERATOFORM, INC. (US) 1999-08-05 WO disclosed