SCHEMBL6067666

SCHEMBL6067666

CC(C=Cc1ccccc1)(C(=O)O)C(=O)O

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.67
EGFR P00533 1/20 0.50
GLA P06280 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
HDAC1 Q13547 3/20 0.48
LMNA P02545 3/20 0.48
HDAC3 O15379 2/20 0.48
HDAC4 P56524 2/20 0.48
HDAC2 Q92769 2/20 0.48
HDAC8 Q9BY41 2/20 0.48
HDAC6 Q9UBN7 2/20 0.48
PLIN1 O60240 2/20 0.48
MAPT P10636 2/20 0.48
RECQL P46063 2/20 0.48
PLIN5 Q00G26 2/20 0.48
ABHD5 Q8WTS1 2/20 0.48
ALDH1A1 P00352 2/20 0.48
TNKS O95271 1/20 0.48
HCAR2 Q8TDS4 1/20 0.48
HDAC7 Q8WUI4 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6067715 0.89 CYP2C19 (0.54) CYP2C19EGFRGLATDP1HDAC1
SCHEMBL6693532 0.84 CA12 (0.52) CYP2C19MAPTALDH1A1HCAR2CYP2D6
SCHEMBL28748361 0.83 CYP2C19 (0.67) CYP2C19EGFRGLATDP1HDAC1
SCHEMBL8736402 0.82 LCK (0.50) CYP2C19MAOB
SCHEMBL3508677 0.80 THRB (0.59) CYP2C19HDAC1LMNAHDAC3HDAC2
SCHEMBL10332365 0.79 CYP2C19 (0.61) CYP2C19EGFRGLATDP1HDAC1
SCHEMBL6067649 0.77 MEN1 (0.50) CYP2C19LMNAMAPTRECQLALDH1A1
SCHEMBL20346330 0.77 MEN1 (0.50) CYP2C19LMNAMAPTRECQLALDH1A1
SCHEMBL1618355 0.77 CYP2C19 (0.58) CYP2C19EGFRGLATDP1HDAC1
SCHEMBL23064568 0.76 CYP2C19 (0.62) CYP2C19EGFRGLATDP1HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006100606-A2 PREPARATION OF BETA-AMINO ACID PRECURSORS VIA INDIUM (III) MEDIATED MARKOVNIKOV ADDITION AND KNOEVENAGEL CONDENSATION WARNER-LAMBERT COMPANY LLC (US) 2006-09-28 WO claimed
WO-2006100606-A2 PREPARATION OF BETA-AMINO ACID PRECURSORS VIA INDIUM (III) MEDIATED MARKOVNIKOV ADDITION AND KNOEVENAGEL CONDENSATION WARNER-LAMBERT COMPANY LLC (US) 2006-09-28 WO disclosed