SCHEMBL6071737

SCHEMBL6071737

CCOc1cc2c(c3c1OC(C)(C)C3)C(c1ccc(CC(=O)O)cc1)=NC(C)(C)C2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SSTR5 P35346 2/20 0.41
RXRA P19793 2/20 0.39
RXRB P28702 2/20 0.39
RXRG P48443 2/20 0.39
FFAR4 Q5NUL3 5/20 0.34
CYP26A1 O43174 1/20 0.33
CYP26B1 Q9NR63 1/20 0.33
ALDH1A1 P00352 2/20 0.32
THRB P10828 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
DGAT1 O75907 1/20 0.32
PTGER4 P35408 2/20 0.32
PTPN1 P18031 1/20 0.32
PTPN6 P29350 1/20 0.32
PTPN11 Q06124 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MAPT P10636 1/20 0.32
HTT P42858 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6072329 0.91 ALDH1A1 (0.35) SSTR5FFAR4ALDH1A1THRBL3MBTL1
SCHEMBL6072465 0.91 SSTR5 (0.39) SSTR5FFAR4L3MBTL1MAPT
SCHEMBL6071725 0.90 FFAR4 (0.33) SSTR5FFAR4ALDH1A1KDM4E
Hydrochloric Acid SCHEMBL6071935 0.89 SSTR5 (0.34) SSTR5FFAR4ALDH1A1KDM4E
SCHEMBL6071457 0.89 SSTR5 (0.38) SSTR5FFAR4
SCHEMBL6071755 0.88 KDM4E (0.40) FFAR4ALDH1A1L3MBTL1KDM4EMAPT
Hydrochloric Acid SCHEMBL5784450 0.88 SSTR5 (0.39) SSTR5RXRARXRB
Hydrochloric Acid SCHEMBL6072535 0.88 KDM4E (0.39) FFAR4ALDH1A1L3MBTL1KDM4EMAPT
SCHEMBL6072463 0.88 FFAR4 (0.32) SSTR5FFAR4MAPT
SCHEMBL6071698 0.87 SSTR5 (0.33) SSTR5FFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060106048-A1 Furoisoquinoline derivative and use thereof PASCALI, PETROS P. (CY) 2006-05-18 US disclosed
EP-1541576-A1 FUROISOQUINOLINE DERIVATIVE AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2005-06-15 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060106048-A1 Furoisoquinoline derivative and use thereof PDE3B, PDE2A, PDE3A SSTR5 837/4885RXRA 692/4885RXRB 379/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.