SCHEMBL6072465

SCHEMBL6072465

CCOc1cc2c(c3c1OC(C)(C)C3)C(c1ccc(CCC(=O)O)cc1)=NC(C)(C)C2

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SSTR5 P35346 2/20 0.39
FFAR4 Q5NUL3 6/20 0.37
S1PR1 P21453 2/20 0.35
TP53 P04637 1/20 0.34
MDM2 Q00987 1/20 0.34
MAPT P10636 4/20 0.34
FFAR1 O14842 2/20 0.34
S1PR3 Q99500 1/20 0.34
S1PR5 Q9H228 1/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
LMNA P02545 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6072275 0.91 CYP4F2 (0.36) SSTR5FFAR4MAPTPOLB
SCHEMBL6071737 0.91 SSTR5 (0.41) SSTR5FFAR4MAPTL3MBTL1
SCHEMBL6071725 0.88 FFAR4 (0.33) SSTR5FFAR4NPC1RAB9APOLB
Hydrochloric Acid SCHEMBL6071935 0.87 SSTR5 (0.34) SSTR5FFAR4NPC1RAB9A
SCHEMBL6071457 0.87 SSTR5 (0.38) SSTR5FFAR4S1PR1S1PR3
SCHEMBL6071755 0.87 KDM4E (0.40) FFAR4MAPTFFAR1L3MBTL1POLB
Hydrochloric Acid SCHEMBL5784450 0.86 SSTR5 (0.39) SSTR5
SCHEMBL6072329 0.86 ALDH1A1 (0.35) SSTR5FFAR4MAPTNPC1L3MBTL1
Hydrochloric Acid SCHEMBL6072535 0.86 KDM4E (0.39) FFAR4MAPTFFAR1L3MBTL1POLB
SCHEMBL6072463 0.86 FFAR4 (0.32) SSTR5FFAR4MAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060106048-A1 Furoisoquinoline derivative and use thereof PASCALI, PETROS P. (CY) 2006-05-18 US disclosed
EP-1541576-A1 FUROISOQUINOLINE DERIVATIVE AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2005-06-15 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060106048-A1 Furoisoquinoline derivative and use thereof PDE3B, PDE2A, PDE3A SSTR5 837/4885FFAR4 272/4885S1PR1 1302/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.