SCHEMBL6073329

SCHEMBL6073329

CCCOCC(=O)Nc1cc(Br)cnc1N

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.39
HPGD P15428 1/20 0.39
KDM4E B2RXH2 3/20 0.37
HSD17B10 Q99714 2/20 0.36
KMT2A Q03164 3/20 0.36
RAB9A P51151 2/20 0.36
LMNA P02545 2/20 0.36
MEN1 O00255 1/20 0.36
MAPT P10636 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
HDAC4 P56524 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6073629 0.90 ALDH1A1 (0.49) ALDH1A1HPGDKDM4EHSD17B10KMT2A
SCHEMBL20266375 0.84 HPGD (0.48) ALDH1A1HPGDKMT2ALMNACYP2C19
SCHEMBL30676150 0.84 HPGD (0.48) ALDH1A1HPGDKMT2ALMNACYP2C19
SCHEMBL20703988 0.82 RAB9A (0.46) ALDH1A1HPGDKMT2ARAB9ALMNA
SCHEMBL6073244 0.81 NPSR1 (0.37) KMT2ALMNAMEN1MAPTCYP1A2
SCHEMBL2756208 0.80 CNR2 (0.43) ALDH1A1HPGDKDM4EKMT2ARAB9A
SCHEMBL15713808 0.78 CNR2 (0.42) ALDH1A1HPGDKDM4EKMT2ARAB9A
SCHEMBL1585857 0.76 CYP1A2 (0.48) ALDH1A1HPGDKDM4EHSD17B10CYP1A2
SCHEMBL8253940 0.76 KMT2A (0.39) ALDH1A1KDM4EHSD17B10KMT2AMEN1
SCHEMBL25299222 0.76 KMT2A (0.47) ALDH1A1KDM4EHSD17B10KMT2ARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006126081-A2 PYRIDINO [2 , 3-B] PYRAZINONES AS PDE-5 INHIBITORS PHARMACIA & UPJOHN COMPANY LLC (US) 2006-11-30 WO disclosed
WO-2006126081-A2 PYRIDINO [2 , 3-B] PYRAZINONES AS PDE-5 INHIBITORS PHARMACIA & UPJOHN COMPANY LLC (US) 2006-11-30 WO disclosed