SCHEMBL6076770

SCHEMBL6076770

O=C(O)C1=C(O)C(=O)N(CCN2CCN(C(=O)c3ccccc3)CC2)C1

nearest known ligand 0.59

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.53
MEN1 O00255 3/20 0.53
KCNH2 Q12809 1/20 0.53
KCNA5 P22460 3/20 0.50
DRD2 P14416 2/20 0.50
SIGMAR1 Q99720 1/20 0.50
HTR2A P28223 1/20 0.50
ALDH1A1 P00352 3/20 0.47
KDM4E B2RXH2 1/20 0.47
DRD3 P35462 2/20 0.46
HPGD P15428 1/20 0.46
ALOX15 P16050 1/20 0.45
TSHR P16473 1/20 0.45
HSD17B10 Q99714 1/20 0.45
USP2 O75604 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6077954 0.90 KCNH2 (0.47) KCNH2ALDH1A1KDM4E
SCHEMBL6076762 0.90 KCNA5 (0.51) KMT2AMEN1KCNA5ALDH1A1KDM4E
SCHEMBL6078272 0.84 L3MBTL1 (0.53) DRD2HTR2AALDH1A1KDM4ETSHR
SCHEMBL6076788 0.80 LIPG (0.39) KMT2AMEN1KCNH2ALDH1A1ALOX15
SCHEMBL6077393 0.79 LIPG (0.39) KCNH2DRD2SIGMAR1ALDH1A1KDM4E
SCHEMBL6078249 0.79 PARP1 (0.45) KMT2ADRD2ALDH1A1DRD3
SCHEMBL6077535 0.76 LIPG (0.51) KMT2AALDH1A1KDM4EALOX15HSD17B10
SCHEMBL14366509 0.75 KMT2A (0.71) KMT2AMEN1KCNH2KCNA5DRD2
SCHEMBL7634958 0.75 KMT2A (0.71) KMT2AMEN1KCNH2KCNA5DRD2
SCHEMBL6078320 0.75 LIPG (0.38) SIGMAR1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7109186-B2 4-hydroxy-5-oxo-1-(2-[4-methylpiperazin-1-yl]ethyl)-2,5-dihydro-1H-pyrrole-3-carboxylic acid (3,4-dichlorobenzyl)-methyl-amide for human immunodeficiency virus (HIV) treatment BRISTOL-MYERS SQUIBB COMPANY (US) 2006-09-19 US disclosed
US-20040110804-A1 HIV integrase inhibitors BRISTOL-MYERS SQUIBB COMPANY 2004-06-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040110804-A1 HIV integrase inhibitors CDKN1A, SAMHD1, CTCF KMT2A 736/4885MEN1 4784/4885KCNH2 4138/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.