SCHEMBL6077828

SCHEMBL6077828

CCC(CCN(CC(C)(C)C)C(=O)O)Oc1nc(C(F)(F)F)ccc1C#N

nearest known ligand 0.47

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 2/20 0.47
NOS2 P35228 2/20 0.47
KDM4E B2RXH2 2/20 0.33
TRPV1 Q8NER1 2/20 0.33
MAPT P10636 1/20 0.33
HTT P42858 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
GPR119 Q8TDV5 1/20 0.32
ALDH1A1 P00352 3/20 0.31
PGR P06401 1/20 0.31
AR P10275 1/20 0.31
P2RY12 Q9H244 5/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6077823 0.81 SLC6A4 (0.44) SLC6A4NOS2TRPV1GPR119PGR
SCHEMBL2529368 0.79 SLC6A4 (0.54) SLC6A4NOS2KDM4ETRPV1GPR119
SCHEMBL6077819 0.78 SLC6A4 (0.47) SLC6A4NOS2KDM4ETRPV1MAPT
SCHEMBL6078861 0.75 SLC6A4 (0.52) SLC6A4NOS2KDM4ETRPV1HTT
SCHEMBL6082710 0.75 SLC6A4 (0.46) SLC6A4NOS2GPR119PGRAR
Hydrochloric Acid SCHEMBL6079500 0.74 SLC6A4 (0.53) SLC6A4NOS2KDM4ETRPV1HTT
SCHEMBL2532516 0.74 SLC6A4 (0.55) SLC6A4NOS2KDM4ETRPV1MAPT
SCHEMBL2529137 0.73 SLC6A4 (0.53) SLC6A4NOS2TRPV1MAPTGPR119
SCHEMBL6078728 0.70 SLC6A4 (0.45) SLC6A4NOS2GPR119PGRAR
SCHEMBL6078732 0.70 SLC6A4 (0.45) SLC6A4NOS2GPR119PGRAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7119109-B2 Heteroarylheteroalkylamine derivatives and their use as inhibitors of nitric oxide synthase ASTRAZENECA AB (SE) 2006-10-10 US disclosed
US-20040220234-A1 Heteroarylheteroalkylamine derivatives and their use as inhibitors of nitric oxide synthase ASTRAZENECA AB (SE) 2004-11-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040220234-A1 Heteroarylheteroalkylamine derivatives and their use as inhibitors of nitric oxide synthase NOS3, NOS2, NOS1 SLC6A4 1543/4885NOS2 2/4885KDM4E 1533/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.