SCHEMBL6078876

SCHEMBL6078876

NS(=O)(=O)c1cccc(NS(=O)(=O)c2cc(O)c3ccc(NC(=S)Nc4ccc5ccc(S(=O)(=O)Nc6ccc(Cl)c(C(=O)O)c6)cc5c4)cc3c2)c1

nearest known ligand 0.66

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
ALDH1A1 P00352 1/20 0.48
CA1 P00915 4/20 0.47
CA2 P00918 4/20 0.47
CA9 Q16790 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6078568 0.94 MEN1 (0.48) MEN1KMT2AALDH1A1
SCHEMBL6079442 0.93 MEN1 (0.50) MEN1KMT2AALDH1A1CA1CA2
SCHEMBL6078719 0.93 MEN1 (0.55) MEN1KMT2AALDH1A1CA1CA2
SCHEMBL6079082 0.91 LMNA (0.48) MEN1KMT2AALDH1A1CA1CA2
SCHEMBL6079055 0.87 PRMT1 (0.53) MEN1KMT2AALDH1A1
SCHEMBL6078658 0.86 MEN1 (0.57) MEN1KMT2AALDH1A1CA1CA2
SCHEMBL6079588 0.85 LMNA (0.49) MEN1KMT2AALDH1A1
SCHEMBL6079074 0.84 LMNA (0.54) MEN1KMT2AALDH1A1CA1CA2
SCHEMBL6079368 0.82 MEN1 (0.71) MEN1KMT2AALDH1A1CA1CA2
SCHEMBL6079497 0.82 MEN1 (0.55) MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7071231-B2 Naphthalene ureas as glucose uptake enhancers TELIK, INC. (US) 2006-07-04 US disclosed
US-6458998-B1 NAPHTHALENEUREAS AS ANTIDIABETIC AGENTS TELIK, INC. 2002-10-01 US disclosed