SCHEMBL6079170

SCHEMBL6079170

Cc1cccc(NS(=O)(=O)c2ccc3ccc(NC(=O)Nc4ccc5ccc(S(=O)(=O)Nc6ccc(Cl)c(C(=O)O)c6)cc5c4)cc3c2)c1

nearest known ligand 0.82

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.57
KMT2A Q03164 4/20 0.57
MAPT P10636 2/20 0.56
ALDH1A1 P00352 2/20 0.52
IDH1 O75874 1/20 0.51
CRHBP P24387 1/20 0.51
CRHR2 Q13324 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
GHSR Q92847 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6079497 0.92 MEN1 (0.55) MEN1KMT2AMAPTALDH1A1CRHBP
SCHEMBL6079248 0.91 MEN1 (0.58) MEN1KMT2AALDH1A1
SCHEMBL6077690 0.89 MEN1 (0.74) MEN1KMT2A
SCHEMBL6078658 0.87 MEN1 (0.57) MEN1KMT2AMAPTALDH1A1
SCHEMBL6429403 0.86 LMNA (0.62) MEN1KMT2AMAPTALDH1A1SMN1; SMN2
SCHEMBL6079195 0.85 TP53 (0.60) MEN1KMT2AALDH1A1
SCHEMBL6078214 0.85 MEN1 (0.57) MEN1KMT2AALDH1A1
SCHEMBL6078607 0.84 MEN1 (0.53) MEN1KMT2AALDH1A1
SCHEMBL6078679 0.83 LMNA (0.56) MEN1KMT2AMAPTALDH1A1CRHBP
SCHEMBL6079356 0.82 MEN1 (0.56) MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7071231-B2 Naphthalene ureas as glucose uptake enhancers TELIK, INC. (US) 2006-07-04 US disclosed
EP-1181271-B1 NAPHTHALENE UREAS AS GLUCOSE UPTAKE ENHANCERS TELIK INC (US) 2005-01-19 EP disclosed
US-6458998-B1 NAPHTHALENEUREAS AS ANTIDIABETIC AGENTS TELIK, INC. 2002-10-01 US disclosed