SCHEMBL6079374

SCHEMBL6079374

Cc1noc(C)c1S(=O)(=O)NC(=O)CCCN1CC(C(=O)O)=C(O)C1=O

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.38
TSHR P16473 2/20 0.38
HPGD P15428 2/20 0.36
HTT P42858 2/20 0.36
GFER P55789 1/20 0.35
CCR1 P32246 1/20 0.35
LIPG Q9Y5X9 1/20 0.35
NPSR1 Q6W5P4 1/20 0.34
ACLY P53396 1/20 0.34
NR3C1 P04150 1/20 0.33
NR3C2 P08235 1/20 0.33
BCL2 P10415 1/20 0.33
BCL2L1 Q07817 1/20 0.33
LMNA P02545 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.32
KMT2A Q03164 1/20 0.32
PKM P14618 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6078393 0.79 LIPG (0.50) LIPG
SCHEMBL6076742 0.73 LIPG (0.42) LIPG
SCHEMBL6078405 0.68 LIPG (0.38) LIPG
SCHEMBL6078842 0.66 LIPG (0.38) ALDH1A1HTTLIPGLMNA
SCHEMBL6078911 0.64 KMT2A (0.42) ALDH1A1TSHRHPGDHTTLIPG
SCHEMBL6077649 0.62 LIPG (0.38) LIPG
SCHEMBL6076712 0.61 L3MBTL1 (0.38) ALDH1A1TSHRHPGDLIPG
SCHEMBL6077439 0.61 LIPG (0.35) TSHRLIPG
SCHEMBL6077645 0.61 LIPG (0.40) LIPG
SCHEMBL6077755 0.60 LIPG (0.49) ALDH1A1LIPGKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7109186-B2 4-hydroxy-5-oxo-1-(2-[4-methylpiperazin-1-yl]ethyl)-2,5-dihydro-1H-pyrrole-3-carboxylic acid (3,4-dichlorobenzyl)-methyl-amide for human immunodeficiency virus (HIV) treatment BRISTOL-MYERS SQUIBB COMPANY (US) 2006-09-19 US disclosed
US-20040110804-A1 HIV integrase inhibitors BRISTOL-MYERS SQUIBB COMPANY 2004-06-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040110804-A1 HIV integrase inhibitors CDKN1A, SAMHD1, CTCF ALDH1A1 563/4885TSHR 4830/4885HPGD 1650/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.